SCHEMBL6088037

SCHEMBL6088037

Nc1nc(-c2ncccn2)nc2cc[c]cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.41
ADORA1 P30542 2/20 0.41
CYP1A1 P04798 5/20 0.36
CYP1A2 P05177 5/20 0.36
CYP1B1 Q16678 5/20 0.36
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
HK1 P19367 1/20 0.33
HKDC1 Q2TB90 1/20 0.33
DCPS Q96C86 1/20 0.33
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
GLA P06280 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6091929 0.87 ADORA2A (0.38) ADORA2AADORA1CYP1A1CYP1A2CYP1B1
SCHEMBL3820902 0.75 DCPS (0.53) DCPS
SCHEMBL8222632 0.73 ADORA2A (0.35) ADORA2AADORA1RAB9ANPC1HK1
SCHEMBL6090464 0.70 SYK (0.36) ADORA2AADORA1RAB9ANPC1HK1
SCHEMBL2000322 0.68 PI4KA (0.53)
SCHEMBL27924195 0.66 HSP90AA1 (0.41) ADORA2AADORA1RAB9ANPC1KDM4E
SCHEMBL6090261 0.66 ADORA2A (0.44) ADORA2AADORA1CYP1A2RAB9ANPC1
SCHEMBL8219623 0.65 CCR1 (0.42) ADORA2AADORA1CYP1A2RAB9ANPC1
SCHEMBL1996363 0.65 NOS3 (0.53) MAPTF12PLAUNCF1NOS3
SCHEMBL8490190 0.65 NCF1 (0.53) KDM4EALDH1A1LMNATP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005435-B2 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2006-02-28 US disclosed