SCHEMBL6130199

SCHEMBL6130199

COc1cc(P(c2ccccc2)c2ccccc2)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52
TUBB2A Q13885 1/20 0.52
TUBB8 Q3ZCM7 1/20 0.52
TUBA3E Q6PEY2 1/20 0.52
TUBA1A Q71U36 1/20 0.52
TUBA1C Q9BQE3 1/20 0.52
TUBB6 Q9BUF5 1/20 0.52
TUBB2B Q9BVA1 1/20 0.52
TUBB1 Q9H4B7 1/20 0.52
CYP3A4 P08684 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
MAPT P10636 3/20 0.46
MEN1 O00255 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7619968 0.87 ACHE (0.56) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL21980854 0.84 PTGS2 (0.47) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
Bromide SCHEMBL28463593 0.83 PTGS2 (0.46) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL8994697 0.80 TDP1 (0.48) CYP3A4TDP1MEN1MAPK1KMT2A
SCHEMBL1042656 0.78 TUBB4A (0.42) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
Hydrochloric Acid SCHEMBL11656824 0.77 TDP1 (0.44) CYP3A4TDP1MAPTMEN1MAPK1
Methane SCHEMBL660326 0.77 CYP3A4 (0.40) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL19019980 0.76 TNFRSF1A (0.46) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
Methoxymethane SCHEMBL9622762 0.75 CYP3A4 (0.75) CYP3A4TDP1MAPK1SMN1; SMN2ACHE
SCHEMBL17829472 0.74 TDP1 (0.46) CYP3A4TDP1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1341797-A4 ORTHO SUBSTITUTED CHIRAL PHOSPHINES AND PHOSPHINITES AND THEIR USE IN ASYMMETRIC CATAYLTIC REACTIONS PENN STATE RES FOUND (US) 2005-06-15 EP disclosed
US-6855657-B2 Ortho substituted chiral phosphines and phosphinites and their use in asymmetric catalytic reactions THE PENN STATE RESEARCH FOUNDATION (US) 2005-02-15 US disclosed
US-20040068126-A1 Ortho substituted chiral phosphines and phosphinites and their use in asymmetric catalytic reactions THE PENN STATE RESEARCH FOUNDATION 2004-04-08 US disclosed
US-6653485-B2 Particularly effective in Ru-catalyzed asymmetric hydrogenation of beta-ketoesters to beta-hydroxyesters and ruthenium-catalyzed asymmetric hydrogenation of enamides to beta amino acids; catalyst selectivity THE PENN STATE RESEARCH FOUNDATION 2003-11-25 US disclosed
EP-1341797-A1 ORTHO SUBSTITUTED CHIRAL PHOSPHINES AND PHOSPHINITES AND THEIR USE IN ASYMMETRIC CATAYLTIC REACTIONS THE PENN STATE RESEARCH FOUNDATION (US) 2003-09-10 EP disclosed
US-20020128501-A1 Particularly effective in Ru-catalyzed asymmetric hydrogenation of beta-ketoesters to beta-hydroxyesters and ruthenium-catalyzed asymmetric hydrogenation of enamides to beta amino acids; catalyst selectivity THE PENN STATE RESEARCH FOUNDATION 2002-09-12 US disclosed
WO-2002040491-A1 ORTHO SUBSTITUTED CHIRAL PHOSPHINES AND PHOSPHINITES AND THEIR USE IN ASYMMETRIC CATAYLTIC REACTIONS THE PENN STATE RESEARCH FOUNDATION (US) 2002-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040068126-A1 Ortho substituted chiral phosphines and phosphinites and their use in asymmetric catalytic reactions BCKDK, PDK3, HCK TUBB4A 3594/4885TUBB 3112/4885TUBA3C 3814/4885
US-20020128501-A1 Particularly effective in Ru-catalyzed asymmetric hydrogenation of beta-ketoesters to beta-hydroxyesters and ruthenium-catalyzed asymmetric hydrogenation of enamides to beta amino acids; catalyst selectivity HRH4, BCKDK, HRH3 TUBB4A 3655/4885TUBB 3045/4885TUBA3C 3738/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.