SCHEMBL6131836

SCHEMBL6131836

C#CCOc1cc(CN(C)C)ccc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.50
DRD2 P14416 1/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
PDE4B Q07343 2/20 0.43
CA2 P00918 2/20 0.43
ACHE P22303 1/20 0.43
BLM P54132 2/20 0.43
PMP22 Q01453 1/20 0.43
HTR1A P08908 1/20 0.43
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR1E P28566 1/20 0.43
HTR2B P41595 1/20 0.43
HTR3A P46098 1/20 0.43
HTR5A P47898 1/20 0.43
HTR6 P50406 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6131979 0.98 HTR7 (0.49) HTR7DRD2CYP1A2CYP3A4CYP2D6
SCHEMBL29976523 0.84 DRD2 (0.46) DRD2CYP1A2CYP3A4CYP2D6PDE4B
SCHEMBL19806083 0.84 DRD2 (0.46) DRD2CYP1A2CYP3A4CYP2D6PDE4B
SCHEMBL6131791 0.84 KDM4E (0.62) CYP1A2CYP3A4CYP2D6ACHEBLM
SCHEMBL5675706 0.82 HTR7 (0.64) HTR7CYP1A2CYP3A4CYP2D6CA2
SCHEMBL29976179 0.81 PDE4B (0.47) DRD2PDE4BCA2ACHEKDM4E
SCHEMBL19806084 0.81 PDE4B (0.47) DRD2PDE4BCA2ACHEKDM4E
SCHEMBL6131892 0.81 MEN1 (0.67) CYP1A2CYP3A4CYP2D6BLMPMP22
SCHEMBL29975770 0.78 DRD2 (0.52) DRD2CYP1A2CYP3A4CYP2D6PDE4B
SCHEMBL19806087 0.78 DRD2 (0.52) DRD2CYP1A2CYP3A4CYP2D6PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
US-6479495-B1 SIMULTANEOUSLY TREATING DEPRESSION AND MEMORY DYSFUNCTION IN MAMMALS SUFFERING FROM MEMORY DYSFUNCTION AND DEPRESSION AVENTIS PHARMACEUTICALS INC. 2002-11-12 US disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed