SCHEMBL19806084

SCHEMBL19806084

C#CCOc1cc(CO)ccc1OC

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.47
DRD2 P14416 1/20 0.46
CA2 P00918 4/20 0.46
POLB P06746 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
CYP2B6 P20813 1/20 0.45
AR P10275 1/20 0.42
MAOB P27338 2/20 0.41
MAOA P21397 1/20 0.41
HTT P42858 1/20 0.41
CA9 Q16790 3/20 0.41
CA12 O43570 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ATM Q13315 1/20 0.41
CA1 P00915 2/20 0.41
FYN P06241 1/20 0.41
ACHE P22303 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29976179 1.00 PDE4B (0.47) PDE4BDRD2CA2POLBNPC1
SCHEMBL19806086 0.94 POLB (0.52) PDE4BDRD2CA2POLBNPC1
SCHEMBL13438449 0.84 DRD2 (0.46) PDE4BDRD2CA2POLBNPC1
SCHEMBL1890562 0.84 DRD2 (0.46) PDE4BDRD2CA2POLBNPC1
SCHEMBL29976523 0.84 DRD2 (0.46) PDE4BDRD2CA2POLBCYP2B6
SCHEMBL19806083 0.84 DRD2 (0.46) PDE4BDRD2CA2POLBCYP2B6
SCHEMBL19640054 0.82 CYP4F2 (0.56) PDE4BRAB9ACYP2B6HTTKDM4E
SCHEMBL6131836 0.81 HTR7 (0.50) PDE4BDRD2CA2CYP2B6MAOB
SCHEMBL29997296 0.80 CA2 (0.68) CA2POLBNPC1RAB9ACA9
SCHEMBL28170408 0.80 CA2 (0.68) CA2POLBNPC1RAB9ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11725000-B2 Apoptosis inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2023-08-15 US disclosed
US-11725000-B2 Apoptosis inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2023-08-15 US disclosed
US-11725000-B2 Apoptosis inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2023-08-15 US disclosed
CN-110023292-B Apoptosis inhibitors 北京生命科学研究所 2022-10-04 CN disclosed
US-20210309647-A1 Apoptosis Inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-10-07 US disclosed
US-20210309647-A1 Apoptosis Inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-10-07 US disclosed
US-11034680-B2 Apoptosis inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-06-15 US disclosed
US-11034680-B2 Apoptosis inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-06-15 US disclosed
EP-3484854-B1 APOPTOSIS INHIBITORS NAT INSTITUTE OF BIOLOGICAL SCIENCES BEIJING (CN) 2021-01-20 EP disclosed
EP-3484854-B1 APOPTOSIS INHIBITORS NAT INSTITUTE OF BIOLOGICAL SCIENCES BEIJING (CN) 2021-01-20 EP disclosed
US-20190152960-A1 Apoptosis Inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2019-05-23 US disclosed
US-20190152960-A1 Apoptosis Inhibitors NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2019-05-23 US disclosed
WO-2018014802-A1 APOPTOSIS INHIBITORS NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2018-01-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190152960-A1 Apoptosis Inhibitors BAX, SDHA, SDHB PDE4B 2935/4885DRD2 4721/4885CA2 903/4885
US-11725000-B2 Apoptosis inhibitors BAX, SDHA, SDHB PDE4B 2935/4885DRD2 4721/4885CA2 903/4885
US-11034680-B2 Apoptosis inhibitors BAX, SDHA, SDHB PDE4B 2935/4885DRD2 4721/4885CA2 903/4885
US-20210309647-A1 Apoptosis Inhibitors BAX, SDHA, SDHB PDE4B 2935/4885DRD2 4721/4885CA2 903/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.