Quipazine

Quipazine

SCHEMBL6131841

COc1cc(CCO)ccc1O.c1ccc2nc(N3CCNCC3)ccc2c1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.55
HTR3E A5X5Y0 3/20 0.55
HTR3B O95264 3/20 0.55
HTR3A P46098 3/20 0.55
HTR3D Q70Z44 3/20 0.55
HTR3C Q8WXA8 3/20 0.55
CYP3A4 P08684 2/20 0.55
HSD17B10 Q99714 2/20 0.55
ALDH1A1 P00352 2/20 0.55
CYP1A2 P05177 2/20 0.55
USP2 O75604 1/20 0.55
ADRB1 P08588 1/20 0.55
HTR1A P08908 1/20 0.55
HTR2C P28335 1/20 0.55
MAPK1 P28482 1/20 0.55
SLC6A4 P31645 1/20 0.55
HTR7 P34969 1/20 0.55
HTT P42858 1/20 0.55
HTR6 P50406 1/20 0.55
PMP22 Q01453 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131974 0.83 NPC1 (0.54) KDM4EHTR3EHTR3BHTR3AHTR3D
SCHEMBL6131873 0.83 ALDH1A1 (0.53) KDM4EHSD17B10ALDH1A1HTR1AMAPK1
SCHEMBL6131972 0.79 TMEM97 (0.56) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL6132097 0.78 TMEM97 (0.55) KDM4EHTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL6131880 0.77 TMEM97 (0.55) KDM4EHTR3EHTR3BHTR3AHTR3D
SCHEMBL6131864 0.76 ADRA1D (0.56) KDM4EHTR3EHTR3BHTR3AHTR3D
Quipazine SCHEMBL322181 0.74 KDM4E (1.00) KDM4EHTR3EHTR3BHTR3AHTR3D
Quipazine SCHEMBL4062074 0.73 KDM4E (0.97) KDM4EHTR3EHTR3BHTR3AHTR3D
SCHEMBL6131973 0.71 HRH3 (0.56) KDM4EHTR3EHTR3BHTR3AHTR3D
SCHEMBL30045575 0.71 TAAR1 (0.73) KDM4ECYP3A4ALDH1A1MAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed