SCHEMBL6131873

SCHEMBL6131873

COc1cc(CCO)ccc1O.c1ccc(N2CCNCC2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.53
KDM4E B2RXH2 5/20 0.53
HPGD P15428 4/20 0.53
HSD17B10 Q99714 4/20 0.53
PLD1 Q13393 1/20 0.52
TMEM97 Q5BJF2 2/20 0.48
TSHR P16473 4/20 0.47
MAPK1 P28482 3/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HTR1A P08908 1/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quipazine SCHEMBL6131841 0.83 KDM4E (0.55) ALDH1A1KDM4EHSD17B10TMEM97MAPK1
SCHEMBL6131854 0.82 HTR1A (0.58) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL6131972 0.81 TMEM97 (0.56) TMEM97TSHRMAPK1LMNAMAPT
SCHEMBL6131864 0.80 ADRA1D (0.56) ALDH1A1KDM4EHSD17B10TMEM97TSHR
Hydrochloric Acid SCHEMBL6132097 0.80 TMEM97 (0.55) ALDH1A1KDM4ETMEM97TSHRMAPK1
SCHEMBL6131990 0.79 ALDH1A1 (0.71) ALDH1A1KDM4EHPGDHSD17B10TSHR
Hydrochloric Acid SCHEMBL6131880 0.79 TMEM97 (0.55) ALDH1A1KDM4ETMEM97TSHRMAPK1
Hydrochloric Acid SCHEMBL6131775 0.78 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL30045575 0.74 TAAR1 (0.73) ALDH1A1KDM4ETSHRMAPK1LMNA
SCHEMBL43681 0.74 TAAR1 (0.73) ALDH1A1KDM4ETSHRMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed