SCHEMBL6131881

SCHEMBL6131881

COc1ccc(CCN2CCN(c3ccccn3)CC2)cc1F

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.58
ALDH1A1 P00352 3/20 0.57
KDM4E B2RXH2 2/20 0.57
LMNA P02545 1/20 0.57
TSHR P16473 1/20 0.57
MAPK1 P28482 1/20 0.57
HTT P42858 1/20 0.57
DRD2 P14416 2/20 0.56
DRD4 P21917 2/20 0.56
HTR2A P28223 2/20 0.56
HTR7 P34969 2/20 0.56
DRD3 P35462 2/20 0.56
ADRA2C P18825 1/20 0.56
DRD1 P21728 1/20 0.56
DRD5 P21918 1/20 0.56
HRH1 P35367 1/20 0.56
ADRA1D P25100 3/20 0.54
ADRA1A P35348 3/20 0.54
ADRA1B P35368 3/20 0.54
HPGD P15428 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6131899 0.99 HTR1A (0.57) HTR1AALDH1A1KDM4ELMNATSHR
SCHEMBL6131854 0.84 HTR1A (0.58) HTR1AALDH1A1KDM4ELMNATSHR
SCHEMBL6131831 0.84 HTR1A (0.50) HTR1AALDH1A1KDM4ELMNADRD2
SCHEMBL6131982 0.83 HTR1A (0.59) HTR1ALMNADRD2DRD4HTR2A
Hydrochloric Acid SCHEMBL6131783 0.81 HTR1A (0.57) HTR1ALMNADRD2DRD4HTR2A
SCHEMBL6131908 0.80 ALDH1A1 (0.58) HTR1AALDH1A1KDM4ELMNATSHR
Hydrochloric Acid SCHEMBL6132036 0.79 ALDH1A1 (0.57) HTR1AALDH1A1KDM4ELMNATSHR
Oxalic Acid SCHEMBL9077864 0.79 SIGMAR1 (0.74) ALDH1A1KDM4ELMNATSHRMAPK1
SCHEMBL6132048 0.77 ALDH1A1 (0.57) HTR1AALDH1A1KDM4ELMNATSHR
Hydrochloric Acid SCHEMBL6131914 0.76 ALDH1A1 (0.56) HTR1AALDH1A1KDM4ELMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP claimed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP claimed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO claimed