SCHEMBL6131922

SCHEMBL6131922

COc1ccc(C(=O)c2ccccc2)cc1F

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.71
LMNA P02545 3/20 0.70
HTT P42858 2/20 0.70
MAPK1 P28482 2/20 0.70
RAB9A P51151 1/20 0.70
CYP1A2 P05177 2/20 0.67
CYP2C19 P33261 2/20 0.67
CYP2D6 P10635 1/20 0.67
HPGD P15428 1/20 0.67
PTGS1 P23219 1/20 0.60
PTGS2 P35354 1/20 0.60
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
TSHR P16473 1/20 0.58
ALDH1A1 P00352 3/20 0.54
GAA P10253 1/20 0.54
L3MBTL1 Q9Y468 3/20 0.53
BCHE P06276 2/20 0.52
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28217099 0.91 HTT (0.76) ACHELMNAHTTMAPK1RAB9A
SCHEMBL7808687 0.88 ACHE (0.77) ACHELMNAHTTMAPK1RAB9A
SCHEMBL11115156 0.88 HTT (0.67) ACHELMNAHTTMAPK1RAB9A
SCHEMBL5520271 0.87 RAB9A (0.61) ACHELMNAHTTMAPK1RAB9A
SCHEMBL27832801 0.87 CYP1A2 (0.62) ACHELMNAHTTMAPK1RAB9A
SCHEMBL6441737 0.87 ALDH1A1 (0.73) ACHELMNAHTTMAPK1RAB9A
SCHEMBL3468365 0.85 HTT (0.63) ACHELMNAHTTMAPK1RAB9A
SCHEMBL3468486 0.85 LMNA (0.63) ACHELMNAHTTMAPK1RAB9A
SCHEMBL31164291 0.85 HTT (0.63) ACHELMNAHTTMAPK1RAB9A
SCHEMBL1443452 0.84 LMNA (0.67) ACHELMNAHTTMAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3994125-B1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMA (US) 2025-12-24 EP disclosed
US-20240299402-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2024-09-12 US disclosed
US-11957687-B2 Modulators of HSD17B13 and methods of use thereof REGENERON PHARMACEUTICALS, INC. (US) 2024-04-16 US disclosed
US-20230094341-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2023-03-30 US disclosed
EP-3994125-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF Regeneron Pharmaceuticals, Inc. (US) 2022-05-11 EP disclosed
WO-2021003295-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed
WO-2021003295-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2021-01-07 WO disclosed
EP-1214310-B1 NOVEL PHOTOCHROMIC NAPHTHOPYRANS TRANSITIONS OPTICAL INC (US) 2005-04-27 EP disclosed
EP-1214310-A1 NOVEL PHOTOCHROMIC NAPHTHOPYRANS TRANSITIONS OPTICAL, INC. (US) 2002-06-19 EP disclosed
US-6348604-B1 COMPOUNDS IN WHICH SELECTION AND PLACEMENT OF SUBSTITUENTS CONTROL WAVELENGTH AND/OR INTENSITY OF VISIBLE ABSORBANCE BANDS PPG INDUSTRIES OHIO, INC. 2002-02-19 US disclosed
WO-2001019812-A1 NOVEL PHOTOCHROMIC NAPHTHOPYRANS TRANSITIONS OPTICAL, INC. (US) 2001-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240299402-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF HSD17B3, HSD17B11, HSD17B1 ACHE 4662/4885LMNA 2981/4885HTT 3611/4885
US-20230094341-A1 MODULATORS OF HSD17B13 AND METHODS OF USE THEREOF HSD17B3, HSD17B11, HSD17B1 ACHE 4662/4885LMNA 2981/4885HTT 3611/4885
US-11957687-B2 Modulators of HSD17B13 and methods of use thereof HSD17B3, HSD17B11, HSD17B1 ACHE 4662/4885LMNA 2981/4885HTT 3611/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.