SCHEMBL6132334

SCHEMBL6132334

COC1(c2ccccc2)CCN(c2ccc(N3CCNCC3)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 7/20 0.54
SIGMAR1 Q99720 6/20 0.54
HTR3E A5X5Y0 5/20 0.54
HTR3B O95264 5/20 0.54
HTR3A P46098 5/20 0.54
HTR3D Q70Z44 5/20 0.54
HTR3C Q8WXA8 5/20 0.54
LTA4H P09960 3/20 0.53
OPRM1 P35372 1/20 0.51
OPRD1 P41143 1/20 0.51
OPRK1 P41145 1/20 0.51
OPRL1 P41146 1/20 0.51
USP2 O75604 2/20 0.50
CYP2D6 P10635 1/20 0.50
HTR6 P50406 3/20 0.47
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HTR5A P47898 1/20 0.43
HTR1A P08908 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6132525 0.86 ADRB1 (0.61) ADRB1SIGMAR1HTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL6132311 0.85 ADRB1 (0.59) ADRB1SIGMAR1HTR3EHTR3BHTR3A
SCHEMBL613551 0.79 OPRM1 (0.55) SIGMAR1OPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL6132329 0.78 OPRM1 (0.47) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL6132476 0.78 USP2 (0.58) OPRM1OPRD1OPRK1OPRL1USP2
Hydrochloric Acid SCHEMBL2420658 0.77 OPRM1 (0.53) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL29638934 0.75 OPRM1 (0.47) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL12122918 0.74 OPRM1 (0.63) OPRM1OPRD1OPRK1OPRL1TSHR
SCHEMBL6132853 0.73 ALDH1A1 (0.53) OPRM1OPRD1OPRK1CYP2D6ALDH1A1
SCHEMBL13876257 0.73 OPRM1 (0.59) OPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884868-B1 Cyclic hexapeptides having antibiotic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-04-26 US disclosed
EP-1173472-A1 CYCLIC HEXAPEPTIDES HAVING ANTIBIOTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-01-23 EP disclosed
WO-2000064927-A1 CYCLIC HEXAPEPTIDES HAVING ANTIBIOTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-11-02 WO disclosed