SCHEMBL6141544

SCHEMBL6141544

O=C(O)c1ccccc1Nc1ccc(C(F)(F)F)cc1[N+](=O)[O-]

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.82
AKR1C2 P52895 5/20 0.82
AKR1B1 P15121 3/20 0.82
AKR1C4 P17516 3/20 0.82
AKR1C1 Q04828 3/20 0.82
KCNMA1 Q12791 1/20 0.62
TAS2R14 Q9NYV8 4/20 0.62
MAPT P10636 6/20 0.56
LMNA P02545 2/20 0.56
HTT P42858 1/20 0.56
MAPK1 P28482 1/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
ALDH1A1 P00352 2/20 0.54
MYC P01106 1/20 0.54
AKR1B10 O60218 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
POLB P06746 1/20 0.53
CCR6 P51684 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141543 1.00 AKR1C3 (0.82) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL6141317 0.87 AKR1C3 (0.63) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL22720171 0.84 TAS2R14 (0.74) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL21248526 0.83 AKR1C3 (0.67) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL9118458 0.83 KCNMA1 (0.66) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL6813056 0.83 TAS2R14 (0.77) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL18667006 0.82 HCAR3 (0.72) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL1688337 0.82 AKR1C3 (0.69) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL13811262 0.81 MAPK1 (0.75) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL16737110 0.81 AKR1C3 (0.71) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1525183-A1 INHIBITORS OF HCV NS5B POLYMERASE Pharmacia & Upjohn Company LLC (US) 2005-04-27 EP disclosed
WO-2004002940-A1 INHIBITORS OF HCV NS5B POLYMERASE PHARMACIA & UPJOHN COMPANY (US) 2004-01-08 WO disclosed