SCHEMBL6142571

SCHEMBL6142571

NC(N)=Nc1cc2ncccc2cc1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.45
ADRA2B P18089 3/20 0.45
ADRA2C P18825 3/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
HTT P42858 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
CASP6 P55212 1/20 0.41
ALDH1A1 P00352 4/20 0.41
CASP1 P29466 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
CASP7 P55210 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6142181 0.81 PLAU (0.50) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL22324148 0.73 ALDH1A1 (0.53) ADRA1AHTTCYP1A2CYP2C19CASP6
SCHEMBL6142541 0.70 ADRA2A (0.62) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL1163802 0.69 HTT (0.53) HTTCYP1A2CYP2C19CASP6ALDH1A1
SCHEMBL28370443 0.69 CASP6 (0.62) HTTCYP1A2CYP2C19CASP6ALDH1A1
SCHEMBL30540041 0.69 HTT (0.53) HTTCYP1A2CYP2C19CASP6ALDH1A1
SCHEMBL8123144 0.69 ALDH1A1 (0.53) ADRA1AHTTCYP1A2CYP2C19CASP6
SCHEMBL3587363 0.69 ALDH1A1 (0.53) HTTCYP1A2CYP2C19CASP6ALDH1A1
SCHEMBL30456422 0.69 ALDH1A1 (0.53) HTTCYP1A2CYP2C19CASP6ALDH1A1
SCHEMBL150476 0.69 NPC1 (0.65) HTTCYP1A2CYP2C19CASP6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944604-B1 GUANIDINYL HETEROCYCLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS PROCTER & GAMBLE (US) 2005-01-12 EP claimed