SCHEMBL6152396

SCHEMBL6152396

CCOC(=O)COc1ccc(-c2cccc(-c3cc(C)[nH]c3C)n2)c2c1C1CCC2C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
PTPN1 P18031 1/20 0.35
F9 P00740 1/20 0.35
SQOR Q9Y6N5 1/20 0.35
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PDE10A Q9Y233 2/20 0.33
CASP3 P42574 1/20 0.33
CASP7 P55210 1/20 0.33
CASP9 P55211 1/20 0.33
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6153077 0.90 NOS3 (0.46) NOS3NOS1NOS2KDM4E
SCHEMBL6155624 0.88 NOS3 (0.43) NOS3NOS1NOS2
SCHEMBL6152398 0.81 NOS3 (0.45) NOS3NOS1NOS2PTPN1F9
SCHEMBL5833973 0.81 NOS3 (0.42) NOS3NOS1NOS2PTPN1F9
SCHEMBL6152762 0.81 NOS3 (0.46) NOS3NOS1NOS2SMN1; SMN2
SCHEMBL6152658 0.80 NOS3 (0.68) NOS3NOS1NOS2PTPN1ALDH1A1
SCHEMBL6153073 0.70 NOS3 (0.47) NOS3NOS1NOS2ALDH1A1KDM4E
SCHEMBL5833906 0.70 NOS3 (0.44) NOS3NOS1NOS2ALDH1A1KDM4E
Dimethylamine SCHEMBL6153154 0.66 NOS1 (0.69) NOS3NOS1NOS2
SCHEMBL6700485 0.66 MEN1 (0.49) ALDH1A1KDM4ESMN1; SMN2NPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084109-B1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS PFIZER PROD INC (US) 2005-01-26 EP disclosed
EP-1084109-A1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS Pfizer Products Inc. (US) 2001-03-21 EP disclosed
WO-1999062883-A1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NITRIC OXIDE SYNTHASE INHIBITORS PFIZER PRODUCTS INC. (US) 1999-12-09 WO disclosed