SCHEMBL6152469

SCHEMBL6152469

C#CCSc1ccc(OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
CA4 P22748 1/20 0.49
MAOB P27338 2/20 0.47
MAOA P21397 1/20 0.47
APP P05067 1/20 0.47
CA7 P43166 1/20 0.44
CA14 Q9ULX7 1/20 0.44
KDM4E B2RXH2 2/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
PYCR1 P32322 1/20 0.43
PTGS2 P35354 1/20 0.43
DAO P14920 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8127145 0.83 MAOB (0.50) ALDH1A1NPC1SMN1; SMN2CA12CA1
SCHEMBL17041364 0.80 MAOB (0.56) ALDH1A1SMN1; SMN2CA12CA1CA2
SCHEMBL20873387 0.78 MTNR1B (0.49) ALDH1A1NPC1RAB9ASMN1; SMN2CA1
SCHEMBL5178079 0.77 CA12 (0.53) ALDH1A1NPC1RAB9ASMN1; SMN2CA12
SCHEMBL418525 0.76 ALDH1A1 (0.59) ALDH1A1NPC1RAB9ASMN1; SMN2CA12
SCHEMBL10578987 0.76 HTT (0.56) ALDH1A1NPC1RAB9ASMN1; SMN2CA12
SCHEMBL10346038 0.74 RAB9A (0.53) ALDH1A1NPC1RAB9ASMN1; SMN2CA12
SCHEMBL28344902 0.74 CA1 (0.52) ALDH1A1NPC1RAB9ACA12CA1
SCHEMBL1323789 0.74 APP (0.53) ALDH1A1NPC1RAB9ASMN1; SMN2CA12
1,4-Dimethoxybenzene SCHEMBL27368038 0.73 CA1 (0.58) ALDH1A1NPC1RAB9ASMN1; SMN2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563056-B Triazoles for modulating intracellular calcium homeostasis 巴斯克大学 2022-08-16 CN disclosed
US-11377427-B2 Triazoles for regulating intracellular calcium homeostasis UNIVERSIDAD DEL PAIS VASCO (ES) 2022-07-05 US disclosed
EP-3466933-B1 TRIAZOLES FOR REGULATING INTRACELLULAR CALCIUM HOMEOSTASIS UNIV DEL PAIS VASCO/EUSKAL HERRIKO UNIBERTSITATEA (ES) 2020-12-02 EP disclosed
US-20200317625-A1 TRIAZOLES FOR REGULATING INTRACELLULAR CALCIUM HOMEOSTASIS UNIVERSIDAD DEL PAIS VASCO (ES) 2020-10-08 US disclosed
EP-3466933-A1 TRIAZOLES FOR REGULATING INTRACELLULAR CALCIUM HOMEOSTASIS Universidad del Pais Vasco (ES) 2019-04-10 EP disclosed
EP-1334095-B1 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO (JP) 2005-01-19 EP disclosed
EP-1334095-A4 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO (JP) 2004-03-17 EP disclosed
US-6693203-B2 REACTING NOPINONE ENOLATE WITH ALKYL 7-HALO-5-HEPTYNOATE, REACTING PRODUCT WITH HYDROXYLAMINE, TREATING WITH TITANIUM TRICHLORIDE AND BORANE REAGENT, HYDROGENATING, REACTING WITH 5-HYDROXY-4-BENZOTHIOPHENECARBOXYLIC ACID, HYDROLYZING SHIONOGI & CO., LTD (JP) 2004-02-17 US disclosed
US-20030199702-A1 Process for the preparation of pgd2 antagonist LARSEN ROBERT (US) 2003-10-23 US disclosed
EP-1334095-A1 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO., LTD. (JP) 2003-08-13 EP disclosed
WO-2002032892-A1 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO., LTD (JP) 2002-04-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11377427-B2 Triazoles for regulating intracellular calcium homeostasis RYR1, ATP2A3, RYR2 ALDH1A1 3347/4885NPC1 2220/4885RAB9A 1224/4885
US-20200317625-A1 TRIAZOLES FOR REGULATING INTRACELLULAR CALCIUM HOMEOSTASIS RYR1, ATP2A3, RYR2 ALDH1A1 3347/4885NPC1 2220/4885RAB9A 1224/4885
US-20030199702-A1 Process for the preparation of pgd2 antagonist PTGDR, PTGDR2, PTGER2 ALDH1A1 3338/4885NPC1 4429/4885RAB9A 4615/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.