SCHEMBL7450787

SCHEMBL7450787

CN(C)CCOc1ccc(-c2ccccn2)c2c1C1CCC2C1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 6/20 0.71
NOS1 P29475 6/20 0.71
NOS2 P35228 5/20 0.71
HTR7 P34969 3/20 0.43
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ACVR1B P36896 1/20 0.38
TGFBR1 P36897 1/20 0.38
HTR1B P28222 1/20 0.37
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
IGF1R P08069 1/20 0.36
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
CHRM2 P08172 1/20 0.36
PTPN1 P18031 1/20 0.35
ADRA2A P08913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7868256 0.95 NOS3 (0.64) NOS3NOS1NOS2HTR7KDM4E
SCHEMBL5838088 0.83 NOS1 (1.00) NOS3NOS1NOS2
SCHEMBL6152661 0.79 NOS3 (0.71) NOS3NOS1NOS2HTR7KDM4E
SCHEMBL6152658 0.78 NOS3 (0.68) NOS3NOS1NOS2HTR7KDM4E
SCHEMBL6152558 0.78 NOS1 (0.91) NOS3NOS1NOS2
SCHEMBL19154076 0.66 KDM4E (0.53) NOS3NOS1NOS2HTR7KDM4E
SCHEMBL4854673 0.66 ERN1 (0.51) NOS3NOS1NOS2HTR7KDM4E
SCHEMBL23405947 0.66 CHRNB2 (0.54) KDM4ESMN1; SMN2ACVR1BTGFBR1ADRB2
SCHEMBL29743809 0.66 CHRNB2 (0.54) KDM4ESMN1; SMN2ACVR1BTGFBR1ADRB2
SCHEMBL4138229 0.66 CYP2D6 (0.69) ACVR1BTGFBR1ADRB2ADRB1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178784-A1 NEW PHARMACEUTICAL COMBINATIONS FOR NOS INHIBITORS Pfizer Products Inc. (US) 2002-02-13 EP disclosed
WO-2000071107-A2 NEW PHARMACEUTICAL COMBINATIONS FOR NOS INHIBITORS PFIZER PRODUCTS INC. (US) 2000-11-30 WO disclosed