SCHEMBL6152697

SCHEMBL6152697

COc1ccc2scc(C=O)c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.58
ALDH1A1 P00352 7/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 2/20 0.50
ERN1 O75460 2/20 0.49
TRIM24 O15164 1/20 0.49
TYR P14679 1/20 0.49
TRIM33 Q9UPN9 1/20 0.49
MTNR1A P48039 5/20 0.47
MTNR1B P49286 4/20 0.47
PRF1 P14222 1/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4796572 0.87 CYP2A6 (0.51) CYP2A6ALDH1A1CYP1A2CYP2C19ERN1
SCHEMBL23287803 0.79 MTNR1A (0.48) CYP2A6ALDH1A1MTNR1AMTNR1BPRF1
SCHEMBL788146 0.75 CYP2A6 (0.56) CYP2A6ALDH1A1MTNR1AMTNR1BPRF1
SCHEMBL2960090 0.75 CYP2A6 (0.53) CYP2A6ALDH1A1ERN1KDM4EMAPT
SCHEMBL2022637 0.74 CYP2A6 (1.00) CYP2A6ALDH1A1ERN1PRF1MAPT
SCHEMBL5397554 0.74 CYP2A6 (0.64) CYP2A6ALDH1A1ERN1MTNR1AMTNR1B
SCHEMBL19735067 0.74 CYP2A6 (0.64) CYP2A6ALDH1A1ERN1KDM4EMAPT
SCHEMBL7332731 0.74 CYP2A6 (0.64) CYP2A6ALDH1A1CYP1A2CYP2C19ERN1
SCHEMBL5547486 0.74 MTNR1A (0.47) ALDH1A1MTNR1AMTNR1BPRF1KDM4E
SCHEMBL3640233 0.74 CYP2A6 (0.64) CYP2A6ERN1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1334095-B1 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO (JP) 2005-01-19 EP disclosed
US-20040147787-A1 Process for oxidation of alcohols MILLER ROSS A (US) 2004-07-29 US disclosed
EP-1334095-A4 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO (JP) 2004-03-17 EP disclosed
US-6693203-B2 REACTING NOPINONE ENOLATE WITH ALKYL 7-HALO-5-HEPTYNOATE, REACTING PRODUCT WITH HYDROXYLAMINE, TREATING WITH TITANIUM TRICHLORIDE AND BORANE REAGENT, HYDROGENATING, REACTING WITH 5-HYDROXY-4-BENZOTHIOPHENECARBOXYLIC ACID, HYDROLYZING SHIONOGI & CO., LTD (JP) 2004-02-17 US disclosed
US-20030199702-A1 Process for the preparation of pgd2 antagonist LARSEN ROBERT (US) 2003-10-23 US disclosed
EP-1334095-A1 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO., LTD. (JP) 2003-08-13 EP disclosed
WO-2003006435-A1 PROCESS FOR OXIDATION OF ALCOHOLS MERCK & CO., INC. (US) 2003-01-23 WO disclosed
WO-2002032892-A1 PROCESS FOR THE PREPARATION OF PGD2 ANTAGONIST SHIONOGI & CO., LTD (JP) 2002-04-25 WO disclosed
US-5510353-A TREATING IRRITABLE BOWEL SYNDROME, GASTROESOPHAGEAL REFLUX DISEASE, CONSTIPATION, MIGRAINE HEADACHES SANDOZ LTD. (CH) 1996-04-23 US disclosed
EP-0505322-A1 Aminoguanidines SANDOZ LTD. (CH) 1992-09-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040147787-A1 Process for oxidation of alcohols TPO, ADH1C, GPX4 CYP2A6 587/4885ALDH1A1 68/4885CYP1A2 164/4885
US-20030199702-A1 Process for the preparation of pgd2 antagonist PTGDR, PTGDR2, PTGER2 CYP2A6 227/4885ALDH1A1 3338/4885CYP1A2 158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.