SCHEMBL6157563

SCHEMBL6157563

Cc1nc(Cl)nc(N2CCc3ccc(F)cc3C2C)c1C

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
SLC6A4 P31645 1/20 0.32
SCD O00767 6/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160361 0.91 ESR1 (0.34)
SCHEMBL6157859 0.88 HTR2A (0.37) HTR2AHTR2CSLC6A4
SCHEMBL6968163 0.84 DRD1 (0.39) HTR2AHTR2C
SCHEMBL7000740 0.83 DRD1 (0.39)
SCHEMBL6957781 0.83 DRD1 (0.39)
SCHEMBL6995013 0.83 DRD1 (0.39)
SCHEMBL7835940 0.82 MEN1 (0.35) SLC6A4
Hydrochloric Acid SCHEMBL6159808 0.82 MEN1 (0.34) SLC6A4
SCHEMBL6159299 0.81 KMT2A (0.40) HTR2AHTR2C
SCHEMBL6956621 0.81 MAOA (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131312-B1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2005-10-26 EP disclosed
US-6545008-B1 Inhibitory activity against gastric acid secretion YUHAN CORPORATION (KR) 2003-04-08 US disclosed
CN-1326453-A Novel poyrimidine derivatives and process for preparation thereof YUHAN CORP (KR) 2001-12-12 CN disclosed
EP-1131312-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2001-09-12 EP disclosed
WO-2000029403-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2000-05-25 WO disclosed