SCHEMBL6157859

SCHEMBL6157859

Cc1nc(Cl)nc(N2CCc3ccc(Cl)cc3C2C)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.37
HTR2C P28335 6/20 0.37
HTR2B P41595 6/20 0.37
HTR1A P08908 6/20 0.37
SLC6A4 P31645 2/20 0.37
HRH1 P35367 2/20 0.37
KCNH2 Q12809 2/20 0.37
ADRB1 P08588 1/20 0.37
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
CNR1 P21554 1/20 0.37
SLC6A2 P23975 1/20 0.37
DRD3 P35462 6/20 0.32
NOTUM Q6P988 1/20 0.32
SRD5A1 P18405 1/20 0.31
DRD2 P14416 6/20 0.31
FKBP1A P62942 1/20 0.31
HHAT Q5VTY9 1/20 0.31
ASIC3 Q9UHC3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159540 0.90 HTR2A (0.36) HTR2AHTR2CHTR2BNOTUMSRD5A1
SCHEMBL6157563 0.88 HTR2A (0.36) HTR2AHTR2CSLC6A4
SCHEMBL6968163 0.86 DRD1 (0.39) HTR2AHTR2CHTR2BDRD3DRD2
SCHEMBL7000740 0.85 DRD1 (0.39)
SCHEMBL6995013 0.85 DRD1 (0.39)
SCHEMBL6957781 0.85 DRD1 (0.39)
SCHEMBL6956621 0.83 MAOA (0.48) DRD3DRD2
SCHEMBL7823470 0.82 DRD2 (0.35) HTR2AHTR1AADRA2AADRA2BADRA2C
SCHEMBL6160361 0.81 ESR1 (0.34) NOTUMSRD5A1
Hydrochloric Acid SCHEMBL6157964 0.81 KCNH3 (0.36) HTR2AHTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131312-B1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2005-10-26 EP disclosed
CN-1159312-C Novel poyrimidine derivatives and process for preparation thereof ������������ʽ���� 2004-07-28 CN disclosed
US-6545008-B1 Inhibitory activity against gastric acid secretion YUHAN CORPORATION (KR) 2003-04-08 US disclosed
CN-1326453-A Novel poyrimidine derivatives and process for preparation thereof YUHAN CORP (KR) 2001-12-12 CN disclosed
EP-1131312-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2001-09-12 EP disclosed
WO-2000029403-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2000-05-25 WO disclosed