SCHEMBL6157580

SCHEMBL6157580

[CH](c1ccccc1)N(c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RELA Q04206 1/20 0.39
ALDH1A1 P00352 5/20 0.39
MAOB P27338 2/20 0.39
TSHR P16473 1/20 0.39
CYP2A6 P11509 1/20 0.39
TRPM8 Q7Z2W7 2/20 0.39
LMNA P02545 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
NPSR1 Q6W5P4 1/20 0.35
ALOX15 P16050 1/20 0.35
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NFE2L2 Q16236 1/20 0.33
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3275188 0.78 RELA (0.39) RELAALDH1A1MAOBTSHRCYP2A6
SCHEMBL988301 0.74 MAOB (0.48) RELAALDH1A1MAOBTRPM8LMNA
Benzene SCHEMBL6405642 0.74 MAOB (0.48) RELAALDH1A1MAOBTRPM8LMNA
SCHEMBL4444201 0.74 MAOB (0.48) RELAALDH1A1MAOBTRPM8LMNA
SCHEMBL1851187 0.73
SCHEMBL10706531 0.73 ALDH1A1 (0.39) RELAALDH1A1TRPM8L3MBTL1NPSR1
SCHEMBL8848798 0.70 NFE2L2 (0.39) RELAALDH1A1MAOBTSHRCYP2A6
SCHEMBL27457020 0.69 TRPM8 (0.46) ALDH1A1CYP2A6TRPM8LMNANPSR1
SCHEMBL2960795 0.69 MEN1 (0.40) RELAALDH1A1TSHRLMNAL3MBTL1
SCHEMBL9559745 0.69 MAOB (0.41) RELAALDH1A1MAOBTSHRCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501897-A1 METHOD FOR THE PRODUCTION OF PERYLEN-3,4:9,10-TETRACARBOXYLIC ACID DIIMIDES AND PERYLEN-3,4:9,10-TETRACARBOXYLIC ACID DIANHYDRIDE AND NAPHTALENE-1,8-DICARBOXYLIMIDES BASF AKTIENGESELLSCHAFT (DE) 2005-02-02 EP disclosed
WO-2003091345-A1 METHOD FOR THE PRODUCTION OF PERYLEN-3,4:9,10-TETRACARBOXYLIC ACID DIIMIDES AND PERYLEN-3,4:9,10-TETRACARBOXYLIC ACID DIANHYDRIDE AND NAPHTALENE-1,8-DICARBOXYLIMIDES BASF AKTIENGESELLSCHAFT (DE) 2003-11-06 WO disclosed