SCHEMBL6158827

SCHEMBL6158827

O=C1CC(O)CN1Cc1ccc(COc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.53
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
S1PR5 Q9H228 2/20 0.51
MMP13 P45452 1/20 0.51
HRH3 Q9Y5N1 3/20 0.49
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
FFAR1 O14842 1/20 0.43
SPHK2 Q9NRA0 1/20 0.43
SPHK1 Q9NYA1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6157792 0.96 GRM2 (0.58) GRM2NPC1RAB9AS1PR5MMP13
SCHEMBL6157539 0.86 HPGD (0.50) S1PR5MMP13HPGDTSHRTDP1
SCHEMBL6159065 0.86 HPGD (0.50) S1PR5MMP13HPGDTSHRTDP1
SCHEMBL6157546 0.86 HPGD (0.50) S1PR5MMP13HPGDTSHRTDP1
SCHEMBL6158588 0.85 GRM2 (0.54) GRM2NPC1RAB9AS1PR5MMP13
SCHEMBL4925533 0.84 HPGD (0.64) NPC1RAB9AHPGDTSHRHTT
SCHEMBL4922178 0.84 HPGD (0.64) NPC1RAB9AHPGDTSHRHTT
SCHEMBL4922166 0.84 HPGD (0.64) NPC1RAB9AHPGDTSHRHTT
SCHEMBL31190825 0.84 HPGD (0.64) NPC1RAB9AHPGDTSHRHTT
SCHEMBL6162246 0.82 HPGD (0.57) NPC1RAB9AHPGDTSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 GRM2 1327/4885NPC1 1686/4885RAB9A 4194/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 GRM2 1202/4885NPC1 1847/4885RAB9A 4261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.