SCHEMBL6159600

SCHEMBL6159600

O=C1C=CC(=O)N1Cc1ccc(Oc2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 7/20 0.69
GSK3A P49840 3/20 0.69
GSK3B P49841 3/20 0.69
FAAH O00519 3/20 0.66
PTGS1 P23219 1/20 0.54
PTGS2 P35354 1/20 0.54
CHRM5 P08912 1/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
LTA4H P09960 1/20 0.48
F2 P00734 1/20 0.47
PLG P00747 1/20 0.47
ELANE P08246 1/20 0.47
CTSG P08311 1/20 0.47
CMA1 P23946 1/20 0.47
CTRC Q99895 1/20 0.47
FFAR1 O14842 1/20 0.46
CASP3 P42574 1/20 0.45
PTPRF P10586 1/20 0.45
PTPN2 P17706 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25435490 0.82 MGLL (1.00) MGLLGSK3AGSK3BFAAHPTGS1
SCHEMBL207740 0.82 MGLL (1.00) MGLLGSK3AGSK3BFAAHPTGS1
SCHEMBL2570381 0.81 CASP3 (0.63) CHRM5MEN1KMT2ACASP3
SCHEMBL146412 0.80 MGLL (1.00) MGLLGSK3AGSK3BFAAHPTGS1
SCHEMBL22320218 0.79 MGLL (1.00) MGLLGSK3AGSK3BFAAHPTGS1
SCHEMBL6160039 0.78 MEN1 (0.49) MGLLFAAHCHRM5MEN1KMT2A
SCHEMBL3384174 0.78 GSK3A (1.00) MGLLGSK3AGSK3BFAAHCHRM5
SCHEMBL9113591 0.75 MGLL (0.64) MGLLGSK3AGSK3BFAAHPTGS1
SCHEMBL5462796 0.74 GSK3A (0.74) GSK3AGSK3BMEN1KMT2APTPRF
SCHEMBL21215698 0.74 MGLL (0.86) MGLLGSK3AGSK3BFAAHPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 MGLL 4739/4885GSK3A 3511/4885GSK3B 3260/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 MGLL 4776/4885GSK3A 3218/4885GSK3B 2868/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.