SCHEMBL6161473

SCHEMBL6161473

CC(=O)OC1CC(=O)N(Cc2ccc(Oc3ccc(NS(C)(=O)=O)cc3)nc2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
EGLN1 Q9GZT9 9/20 0.36
LTA4H P09960 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
P2RX3 P56373 3/20 0.35
ACACB O00763 2/20 0.35
PGR P06401 1/20 0.34
MMP2 P08253 2/20 0.34
MMP3 P08254 1/20 0.34
MMP9 P14780 1/20 0.34
MMP14 P50281 1/20 0.34
MMP1 P03956 1/20 0.34
ACACA Q13085 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161464 1.00 HCRTR1 (0.36) HCRTR1HCRTR2EGLN1LTA4HHRH3
SCHEMBL6162428 0.86 EGLN1 (0.45) HCRTR1HCRTR2EGLN1P2RX3ACACB
SCHEMBL6162419 0.86 EGLN1 (0.45) HCRTR1HCRTR2EGLN1P2RX3ACACB
SCHEMBL6164470 0.85 EGLN1 (0.44) HCRTR1HCRTR2EGLN1HRH3P2RX3
SCHEMBL6164463 0.85 EGLN1 (0.44) HCRTR1HCRTR2EGLN1HRH3P2RX3
SCHEMBL6161240 0.83 EGLN1 (0.40) HCRTR1HCRTR2EGLN1LTA4HHRH3
SCHEMBL6161230 0.83 EGLN1 (0.40) HCRTR1HCRTR2EGLN1LTA4HHRH3
SCHEMBL6162044 0.78 EGLN1 (0.40) HCRTR1HCRTR2EGLN1LTA4HHRH3
SCHEMBL6159802 0.78 EGLN1 (0.40) HCRTR1HCRTR2EGLN1LTA4HHRH3
SCHEMBL6159586 0.76 LTA4H (0.41) HCRTR1HCRTR2EGLN1LTA4HP2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050165064-A1 Novel thiol derivative, process for producing the same and use thereof TAKEDA PHARMACEUTICALS NORTH AMERICA, INC. 2005-07-28 US disclosed
EP-1500658-A1 NOVEL THIOL DERIVATIVE, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2005-01-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165064-A1 Novel thiol derivative, process for producing the same and use thereof TST, QSOX1, MMP1 HCRTR1 2881/4885HCRTR2 2908/4885EGLN1 841/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.