SCHEMBL6161845

SCHEMBL6161845

FC(F)(F)c1cccc(C2=CCN(CCCCn3cc(Cl)cn3)CC2)c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.54
SIGMAR1 Q99720 4/20 0.43
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
PARP1 P09874 3/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
KCNA3 P22001 1/20 0.39
HTR1A P08908 1/20 0.39
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847491 0.85 SIGMAR1 (0.58) SIGMAR1PARP1HTR1A
SCHEMBL5846299 0.83 SIGMAR1 (0.55) SIGMAR1PARP1HTR1A
SCHEMBL5846267 0.82 SIGMAR1 (0.60) HTR7SIGMAR1PARP1HTR1A
SCHEMBL6162324 0.81 SIGMAR1 (0.57) HTR7SIGMAR1PARP1HTR1A
Hydrochloric Acid SCHEMBL6165778 0.81 SIGMAR1 (0.59) HTR7SIGMAR1PARP1HTR1A
SCHEMBL5848161 0.81 SIGMAR1 (0.60) SIGMAR1PARP1HTR1A
Hydrochloric Acid SCHEMBL7115716 0.80 SIGMAR1 (0.56) HTR7SIGMAR1PARP1HTR1A
SCHEMBL5847759 0.80 SIGMAR1 (0.56) HTR7SIGMAR1PARP1HTR1A
SCHEMBL11269207 0.80 HTR7 (0.60) HTR7SIGMAR1PPARGPPARAPARP1
SCHEMBL6618898 0.79 HTR7 (0.58) HTR7SIGMAR1PPARGPPARAPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721455-B9 TETRAHYDROPYRIDINE-(OR 4-HYDROXYPIPERIDINE)ALKYLAZOLES HAVING AN AFFINITY FOR SIGMA AND/OR 5HT1A RECEPTORS ESTEVE LABOR DR (ES) 2005-04-20 EP claimed
EP-0721455-B1 TETRAHYDROPYRIDINE-(OR 4-HYDROXYPIPERIDINE)ALKYLAZOLES HAVING AN AFFINITY FOR SIGMA AND/OR 5HT1A RECEPTORS ESTEVE LABOR DR (ES) 2002-12-11 EP claimed
US-6232329-B1 POSSESSING THERAPEUTIC ACTIVITY FOR THE TREATMENT OF ANXIETY, PSYCHOSIS, EPILEPSY, CONVULSION, MOTORICITY PROBLEMS, AMNESIA, CEREBROVASCULAR DISEASES OR SENILE DEMENTIA LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2001-05-15 US claimed