SCHEMBL6162216

SCHEMBL6162216

Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CN(C(=O)[C@@H](COCc2ccccc2)NC(=O)C(C)(C)NC(=O)OC(C)(C)C)CC3)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA1 Q09470 4/20 0.48
KCNAB1 Q14722 4/20 0.48
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
P2RX7 Q99572 2/20 0.41
GHSR Q92847 2/20 0.40
PPARA Q07869 1/20 0.39
HCRTR2 O43614 2/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
UGCG Q16739 1/20 0.38
CCKBR P32239 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6164155 0.89 P2RX7 (0.49) KCNA1KCNAB1P2RX7HCRTR2
SCHEMBL6160934 0.89 KCNA1 (0.55) KCNA1KCNAB1MEN1KMT2AGHSR
SCHEMBL6160943 0.89 KCNA1 (0.55) KCNA1KCNAB1MEN1KMT2AGHSR
Hydrochloric Acid SCHEMBL6160591 0.88 KCNA1 (0.55) KCNA1KCNAB1MEN1KMT2AGHSR
Hydrochloric Acid SCHEMBL6160605 0.88 KCNA1 (0.55) KCNA1KCNAB1MEN1KMT2AGHSR
SCHEMBL6162496 0.87 PPARA (0.42) GHSRPPARAHCRTR2CYP3A4UGCG
SCHEMBL6162501 0.87 PPARA (0.42) GHSRPPARAHCRTR2CYP3A4UGCG
SCHEMBL8413200 0.85 PPARA (0.43) GHSRPPARAHCRTR2CCKBRCTSS
SCHEMBL6162692 0.84 NR1H2 (0.48) KMT2AGHSRPPARAHCRTR2CYP3A4
SCHEMBL6162688 0.84 NR1H2 (0.48) KMT2AGHSRPPARAHCRTR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721455-B9 TETRAHYDROPYRIDINE-(OR 4-HYDROXYPIPERIDINE)ALKYLAZOLES HAVING AN AFFINITY FOR SIGMA AND/OR 5HT1A RECEPTORS ESTEVE LABOR DR (ES) 2005-04-20 EP claimed
EP-0721455-B1 TETRAHYDROPYRIDINE-(OR 4-HYDROXYPIPERIDINE)ALKYLAZOLES HAVING AN AFFINITY FOR SIGMA AND/OR 5HT1A RECEPTORS ESTEVE LABOR DR (ES) 2002-12-11 EP claimed
EP-0828754-B1 DIPEPTIDES WHICH PROMOTE RELEASE OF GROWTH HORMONE PFIZER (US) 2005-02-02 EP disclosed