SCHEMBL6163003

SCHEMBL6163003

CC1CC(=O)c2c(CC(C)CC(C)(C)C)nn(-c3ccccc3)c2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 7/20 0.40
CSNK2A2 P19784 5/20 0.40
CSNK2B P67870 5/20 0.40
CSNK2A1 P68400 5/20 0.40
CSNK2A3 Q8NEV1 1/20 0.40
ALDH1A1 P00352 4/20 0.38
TSHR P16473 3/20 0.38
HTT P42858 2/20 0.38
HPGD P15428 2/20 0.38
MAPT P10636 1/20 0.38
BUB1 O43683 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
KHK P50053 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.30
CACNA1H O95180 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6772625 0.90 CSNK2A2 (0.34) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6770294 0.89 SRC (0.36) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6167945 0.88 DHODH (0.37) ABCG2CSNK2A2CSNK2BCSNK2A1ALDH1A1
SCHEMBL6772144 0.87 RIPK2 (0.36) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6167949 0.87 ABCG2 (0.44) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6166197 0.86 CCNA2 (0.41) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6163485 0.83 ALDH1A1 (0.38) ABCG2CSNK2A2CSNK2BCSNK2A1ALDH1A1
SCHEMBL6163506 0.81 CCNA2 (0.35) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6164280 0.81 OPRM1 (0.45) ALDH1A1TSHRHTTLMNAMAPK1
SCHEMBL6168175 0.81 CSNK2A2 (0.33) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed