SCHEMBL6164280

SCHEMBL6164280

CC(Cc1nn(-c2ccccc2)c2c1C(=O)CC(C)(C)C2)CC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 10/20 0.45
ALDH1A1 P00352 5/20 0.42
KMT2A Q03164 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
HSP90AB1 P08238 1/20 0.42
LMNA P02545 4/20 0.42
TSHR P16473 2/20 0.42
SRC P12931 1/20 0.39
HTT P42858 2/20 0.39
HSD17B10 Q99714 2/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6771777 0.90 OPRM1 (0.46) OPRM1ALDH1A1NPSR1HSP90AB1LMNA
SCHEMBL6771450 0.89 OPRM1 (0.46) OPRM1ALDH1A1KMT2ANPSR1HSP90AB1
SCHEMBL6771525 0.87 OPRM1 (0.50) OPRM1ALDH1A1NPSR1HSP90AB1LMNA
SCHEMBL6162256 0.87 OPRM1 (0.50) OPRM1ALDH1A1KMT2ANPSR1HSP90AB1
SCHEMBL6166206 0.86 OPRM1 (0.42) OPRM1ALDH1A1KMT2ANPSR1HSP90AB1
SCHEMBL6163485 0.83 ALDH1A1 (0.38) OPRM1ALDH1A1KMT2ALMNATSHR
SCHEMBL6164838 0.81 CCNA2 (0.41) OPRM1ALDH1A1KMT2ANPSR1HSP90AB1
SCHEMBL6163003 0.81 ABCG2 (0.40) ALDH1A1KMT2ALMNATSHRHTT
SCHEMBL6166030 0.81 ALPL (0.40) OPRM1ALDH1A1KMT2ANPSR1HSP90AB1
SCHEMBL6167945 0.80 DHODH (0.37) ALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed