SCHEMBL6167949

SCHEMBL6167949

CC(C)Cc1nn(-c2ccccc2)c2c1C(=O)CC(C)C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 6/20 0.44
CSNK2A2 P19784 4/20 0.44
CSNK2B P67870 4/20 0.44
CSNK2A1 P68400 4/20 0.44
CSNK2A3 Q8NEV1 1/20 0.44
ALDH1A1 P00352 3/20 0.39
TSHR P16473 2/20 0.39
HTT P42858 2/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
CACNA1H O95180 2/20 0.38
BUB1 O43683 1/20 0.36
CACNA1G O43497 1/20 0.34
KCNH2 Q12809 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
SLC5A1 P13866 2/20 0.33
HIF1A Q16665 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6770545 0.88 ABCG2 (0.38) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6769517 0.88 SRC (0.39) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6162163 0.87 DHODH (0.41) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6163003 0.87 ABCG2 (0.40) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6771827 0.86 ABCG2 (0.37) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6164477 0.84 ABCG2 (0.43) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6165077 0.84 CCNA2 (0.45) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6164455 0.81 ABCG2 (0.47) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL6165127 0.80 ALDH1A1 (0.43) ABCG2CSNK2A2CSNK2BCSNK2A1ALDH1A1
SCHEMBL6167870 0.79 ALDH1A1 (0.49) ABCG2CSNK2A2CSNK2BCSNK2A1CSNK2A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed