SCHEMBL6165864

SCHEMBL6165864

c1cc2c(cc1Oc1ccc3c(c1)OCO3)OCO2

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.78
MAPK1 P28482 1/20 0.78
MAOB P27338 8/20 0.56
CYP3A4 P08684 1/20 0.52
MAOA P21397 4/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
LMNA P02545 3/20 0.51
TP53 P04637 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
GAA P10253 1/20 0.49
MMP13 P45452 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15458939 0.92 ALDH1A1 (0.68) ALDH1A1MAPK1MAOBCYP3A4MAOA
SCHEMBL18415547 0.90 ALDH1A1 (0.71) ALDH1A1MAPK1MAOBMAOANPC1
SCHEMBL7294658 0.88 ALDH1A1 (1.00) ALDH1A1MAPK1MAOBCYP3A4MAOA
SCHEMBL19032000 0.88 ALDH1A1 (0.69) ALDH1A1MAPK1MAOBMAOANPC1
SCHEMBL14743537 0.88 ALDH1A1 (0.69) ALDH1A1MAPK1MAOBCYP3A4MAOA
SCHEMBL257873 0.88 ALDH1A1 (0.69) ALDH1A1MAPK1MAOBNPC1RAB9A
SCHEMBL921951 0.87 ALDH1A1 (0.67) ALDH1A1MAPK1MAOBCYP3A4MAOA
SCHEMBL22162810 0.86 MEN1 (0.64) ALDH1A1MAPK1MAOBCYP3A4MAOA
SCHEMBL16628033 0.84 ALDH1A1 (0.63) ALDH1A1MAPK1MAOBNPC1RAB9A
SCHEMBL9505708 0.84 ALDH1A1 (0.63) ALDH1A1MAPK1MAOBCYP3A4MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113683492-A Preparation method of 3-phenoxybromopropane or analogue thereof 常熟理工学院 2021-11-23 CN disclosed
EP-1102751-A4 NOVEL BI- AND TRI-CYCLIC AZA COMPOUNDS AND THEIR USES UNIV GEORGETOWN (US) 2005-06-22 EP disclosed
US-20040147754-A1 Novel process SMITHKLINE BEECHAM PLC 2004-07-29 US disclosed
US-6716985-B2 ALCOHOLISM, PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 2004-04-06 US disclosed
US-6489347-B1 NOVEL INTERMEDIATE CARBOXALDEHYDES FOR PHARMACEUTICAL PRODUCTS WITH ANTIDEPRESSANT AND ANTI-PARKINSON PROPERTIES SMITHKLINE BEECHAM PLC (GB) 2002-12-03 US disclosed
US-20020133011-A1 Novel process SMITHKLINE BEECHAM PLC 2002-09-19 US disclosed
EP-0986389-A4 NOVEL PROCESS SMITHKLINE BEECHAM CORP (US) 2001-09-12 EP disclosed
EP-1102751-A1 NOVEL BI- AND TRI-CYCLIC AZA COMPOUNDS AND THEIR USES Georgetown University (US) 2001-05-30 EP disclosed
CN-1268889-A Novel process for obtg. intermediates SMITHKLINE BEECHAM CORP (US) 2000-10-04 CN disclosed
EP-0986389-A1 NOVEL PROCESS SMITHKLINE BEECHAM CORPORATION (US) 2000-03-22 EP disclosed
WO-2000007994-A1 NOVEL BI- AND TRI-CYCLIC AZA COMPOUNDS AND THEIR USES GEORGETOWN UNIVERSITY (US) 2000-02-17 WO disclosed
WO-1998053824-A1 NOVEL PROCESS SMITHKLINE BEECHAM CORPORATION (US) 1998-12-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020133011-A1 Novel process HTR1A, HTR4, MAOA ALDH1A1 900/4885MAPK1 2468/4885MAOB 16/4885
US-20040147754-A1 Novel process HTR1A, HTR4, HTR2B ALDH1A1 1013/4885MAPK1 2149/4885MAOB 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.