SCHEMBL6166099

SCHEMBL6166099

O=C1c2ccccc2C(=O)N1CCOCCN1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 6/20 0.79
DRD2 P14416 5/20 0.79
ALDH1A1 P00352 2/20 0.60
GAA P10253 2/20 0.60
POLB P06746 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
LMNA P02545 1/20 0.60
MAPT P10636 1/20 0.60
MAPK1 P28482 1/20 0.60
HRH1 P35367 4/20 0.58
HRH2 P25021 2/20 0.58
HTR2A P28223 2/20 0.58
HTR2B P41595 2/20 0.58
KCNH2 Q12809 2/20 0.58
USP2 O75604 2/20 0.58
ABCB11 O95342 1/20 0.58
CHRM2 P08172 1/20 0.58
ADRA2A P08913 1/20 0.58
ADRA2B P18089 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16757317 0.93 DRD3 (0.81) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL7976323 0.88 DRD2 (0.95) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL9256633 0.88 DRD2 (1.00) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL9733689 0.88 DRD2 (0.84) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL31232750 0.88 DRD2 (0.84) DRD3DRD2ALDH1A1GAAPOLB
Hydrochloric Acid SCHEMBL10826808 0.87 DRD2 (0.92) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL10763449 0.84 DRD2 (0.95) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL9249351 0.81 DRD2 (0.73) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL9257199 0.81 DRD3 (0.86) DRD3DRD2ALDH1A1GAAPOLB
SCHEMBL1463080 0.81 TERT (0.55) DRD3DRD2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060163-B1 NEW PIPERAZINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES KLINGE CO CHEM PHARM FAB (DE) 2005-10-12 EP disclosed
US-6903118-B1 Piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides KLINGE PHARMA GMBH (DE) 2005-06-07 US disclosed
EP-1060163-A1 NEW PIPERAZINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES Klinge Pharma GmbH (DE) 2000-12-20 EP disclosed
WO-1999031063-A1 NEW PIPERAZINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES KLINGE PHARMA GMBH (DE) 1999-06-24 WO disclosed