SCHEMBL6166254

SCHEMBL6166254

N#CCCn1nc(-c2ccco2)c2c1CCC2=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.38
KDM4E B2RXH2 6/20 0.38
HPGD P15428 6/20 0.38
HSD17B10 Q99714 4/20 0.38
MAPT P10636 3/20 0.38
PKM P14618 3/20 0.38
ALOX15 P16050 3/20 0.38
LMNA P02545 3/20 0.38
USP2 O75604 2/20 0.38
TSHR P16473 2/20 0.38
TDP1 Q9NUW8 4/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
POLB P06746 3/20 0.36
ALOX12 P18054 2/20 0.36
CASP1 P29466 2/20 0.36
PTPN7 P35236 2/20 0.36
RECQL P46063 2/20 0.36
BLM P54132 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161914 0.84 HTT (0.44) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL6167558 0.81 BRD4 (0.31) BRD4EP300CREBBP
SCHEMBL6165490 0.78 LMNA (0.49) ALDH1A1HPGDHSD17B10MAPTLMNA
SCHEMBL6167036 0.77 RIPK3 (0.39) ALDH1A1HPGDMAPTKMT2AKDM5A
SCHEMBL6165983 0.77 ATM (0.44) ALDH1A1KDM4EHPGDMAPTTSHR
SCHEMBL6164086 0.76 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL6166453 0.74 ALDH1A1 (0.39) ALDH1A1HPGDHSD17B10MAPTUSP2
SCHEMBL6163581 0.73 CYP1A2 (0.36) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL6165037 0.71 MAOB (0.42) ALDH1A1HSD17B10MAPTALOX15TSHR
SCHEMBL6162649 0.70 PARP1 (0.37) ALDH1A1HSD17B10MAPTALOX15LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed