SCHEMBL6167042

SCHEMBL6167042

COC1CC(C)(C)Cc2c1c(C)nn2-c1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 9/20 0.49
CDK2 P24941 9/20 0.49
ALDH1A1 P00352 6/20 0.45
KDM4E B2RXH2 6/20 0.45
HPGD P15428 5/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CCNO P22674 1/20 0.43
CCNE1 P24864 1/20 0.43
CCNA1 P78396 1/20 0.43
MAPT P10636 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
THRB P10828 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
HSD17B10 Q99714 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165456 0.83 OPRM1 (0.57) CCNA2CDK2ALDH1A1KDM4EHPGD
SCHEMBL6162861 0.71 OPRM1 (0.65) CCNA2CDK2ALDH1A1CCNOCCNE1
SCHEMBL6164586 0.68 LMNA (0.70) CCNA2CDK2ALDH1A1KDM4EHPGD
SCHEMBL6164588 0.68 LMNA (0.70) CCNA2CDK2ALDH1A1KDM4EHPGD
SCHEMBL6163398 0.66 CCNA2 (1.00) CCNA2CDK2CCNOCCNE1CCNA1
SCHEMBL6162155 0.63 OPRM1 (0.57) CCNA2CDK2ALDH1A1KDM4EHPGD
SCHEMBL6167358 0.62 ALDH1A1 (0.57) CCNA2CDK2ALDH1A1KDM4EHPGD
SCHEMBL5235503 0.62 ALDH1A1 (0.43) CCNA2CDK2ALDH1A1KDM4EHPGD
SCHEMBL18949733 0.62 ALDH1A1 (0.55) CCNA2CDK2ALDH1A1KDM4EHPGD
SCHEMBL6164703 0.61 OPRM1 (0.45) CCNA2CDK2ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP claimed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US claimed
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed