SCHEMBL6168330

SCHEMBL6168330

CS(=O)(=O)c1ccccc1C(=O)n1cc(CC(=O)O)c2ccc(Cl)cc21

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.44
AKR1C2 P52895 4/20 0.44
AKR1C4 P17516 1/20 0.44
PTGS1 P23219 1/20 0.44
LMNA P02545 2/20 0.43
ALDH1A1 P00352 1/20 0.43
ABCB1 P08183 2/20 0.42
PTGDR2 Q9Y5Y4 2/20 0.39
HTR6 P50406 3/20 0.38
MCL1 Q07820 2/20 0.37
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7200984 0.81 AKR1C3 (0.56) AKR1C3AKR1C2AKR1C4PTGS1ABCB1
SCHEMBL7202731 0.80 LMNA (0.39) LMNAALDH1A1KMT2A
SCHEMBL28977346 0.76 AKR1C3 (0.49) AKR1C3AKR1C2AKR1C4PTGS1LMNA
SCHEMBL20791852 0.73 ALDH1A1 (0.54) AKR1C3AKR1C2AKR1C4PTGS1LMNA
SCHEMBL6514458 0.71 LMNA (0.49) AKR1C3AKR1C2AKR1C4PTGS1LMNA
SCHEMBL20769675 0.71 AKR1C3 (0.72) AKR1C3AKR1C2AKR1C4PTGS1LMNA
SCHEMBL7208647 0.70 AKR1C3 (0.64) AKR1C3AKR1C2AKR1C4PTGS1LMNA
SCHEMBL6171169 0.70 AKR1C3 (0.46) AKR1C3AKR1C2AKR1C4PTGS1LMNA
SCHEMBL29070101 0.69 ALDH1A1 (0.47) ALDH1A1PTGDR2
SCHEMBL4216463 0.69 AKR1C3 (0.58) AKR1C3AKR1C2AKR1C4PTGS1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045833-B1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2005-11-02 EP disclosed