SCHEMBL6171990

SCHEMBL6171990

CCc1nc2c(OC)ccc(OC(=O)Nc3c(C#N)cnn3C)c2s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
MAPT P10636 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 2/20 0.38
HPGD P15428 4/20 0.37
KDM4E B2RXH2 2/20 0.37
TSHR P16473 2/20 0.37
HSD17B10 Q99714 2/20 0.37
LMNA P02545 2/20 0.37
ADORA2A P29274 3/20 0.36
ADORA2B P29275 3/20 0.36
ADORA1 P30542 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
CACNA1H O95180 1/20 0.35
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
POLB P06746 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6173367 0.82 MAPT (0.48) ALDH1A1MAPTSMN1; SMN2TP53HPGD
SCHEMBL6170768 0.82 TP53 (0.54) ALDH1A1MAPTSMN1; SMN2TP53HPGD
SCHEMBL6170577 0.81 TP53 (0.45) ALDH1A1MAPTSMN1; SMN2TP53HPGD
SCHEMBL6171924 0.79 ADORA2A (0.45) ALDH1A1MAPTSMN1; SMN2HPGDKDM4E
SCHEMBL7470525 0.76 ADORA2A (0.39) MAPTTP53HSD17B10LMNAADORA2A
SCHEMBL6170859 0.72 ALDH1A1 (0.41) ALDH1A1MAPTSMN1; SMN2TP53HPGD
SCHEMBL6612626 0.72 ADORA2A (0.38) ALDH1A1SMN1; SMN2TP53HPGDKDM4E
SCHEMBL6612393 0.72 SMN1; SMN2 (0.36) ALDH1A1SMN1; SMN2TP53HPGDTSHR
SCHEMBL6171107 0.71 ALDH1A1 (0.41) ALDH1A1MAPTSMN1; SMN2TP53HPGD
SCHEMBL7016945 0.68 PDE4A (0.52) ALDH1A1SMN1; SMN2TP53HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263757-B1 BENZTHIAZOLES AS TNF AND PDE-IV INHIBITORS DARWIN DISCOVERY LTD (GB) 2005-07-27 EP claimed