SCHEMBL6173014

SCHEMBL6173014

CC(C)COC(=O)N(C)C[C@@]1(c2ccccc2)C[C@H]1COCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
OPRM1 P35372 2/20 0.34
OPRL1 P41146 2/20 0.34
BCHE P06276 2/20 0.34
ACHE P22303 2/20 0.34
ELANE P08246 1/20 0.34
SLC6A2 P23975 2/20 0.33
CYP3A4 P08684 2/20 0.33
TSHR P16473 2/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CTSL P07711 2/20 0.33
CTSB P07858 2/20 0.33
CTSS P25774 2/20 0.33
CTSK P43235 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171093 1.00 CHRNB2 (0.35) CHRNB2CHRNB4CHRNA3CHRNA4OPRM1
SCHEMBL4028380 0.84 L3MBTL1 (0.43) OPRM1OPRL1SLC6A2SLC6A4SLC6A3
SCHEMBL4029654 0.84 L3MBTL1 (0.43) OPRM1OPRL1SLC6A2SLC6A4SLC6A3
SCHEMBL6172551 0.81 ALDH1A1 (0.39) CYP3A4TSHRALDH1A1CTSLCTSS
SCHEMBL6173847 0.79 LMNA (0.42) CYP3A4TSHRALDH1A1
SCHEMBL4028340 0.75 SLC6A2 (0.41) OPRM1OPRL1SLC6A2TSHRSLC6A4
SCHEMBL4027425 0.75 SLC6A2 (0.41) OPRM1OPRL1SLC6A2TSHRSLC6A4
SCHEMBL4027422 0.75 SLC6A2 (0.41) OPRM1OPRL1SLC6A2TSHRSLC6A4
SCHEMBL4021145 0.73 ALDH1A1 (0.40) OPRM1OPRL1ALDH1A1
SCHEMBL4022452 0.73 ALDH1A1 (0.40) OPRM1OPRL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569934-A2 CYCLOPROPYL COMPOUNDS AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
WO-2004055010-A2 CYCLOPROPYL COMPOUNDS AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed