SCHEMBL6175260

SCHEMBL6175260

CCc1cnccc1C(C)C1NC(=O)N(c2ccc(S(=O)(=O)C(F)(F)F)cc2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 2/20 0.39
LMNA P02545 2/20 0.34
HRH4 Q9H3N8 2/20 0.34
PTGS2 P35354 3/20 0.32
NAMPT P43490 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CTSS P25774 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6173330 0.93 IGF1R (0.40) IGF1RLMNANAMPTMAPK1HTT
SCHEMBL6175529 0.91 IGF1R (0.37) IGF1RLMNAHRH4
SCHEMBL6175175 0.89 IGF1R (0.36) IGF1RLMNAPTGS2MAPK1HTT
SCHEMBL6174640 0.88 IGF1R (0.37) IGF1RLMNAHRH4PTGS2MAPK1
SCHEMBL6171408 0.87 IGF1R (0.35) IGF1RLMNAPTGS2MAPK1HTT
SCHEMBL6176021 0.85 IGF1R (0.34) IGF1RLMNAPTGS2MAPK1HTT
SCHEMBL6175297 0.84 LMNA (0.39) IGF1RLMNAPTGS2MAPK1HTT
SCHEMBL6174658 0.84 RXFP1 (0.34) IGF1RLMNAMAPK1SMN1; SMN2
SCHEMBL6174377 0.83 IGF1R (0.40) IGF1RLMNA
SCHEMBL6174116 0.83 IGF1R (0.33) IGF1RLMNAPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-A2 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-11-30 EP disclosed
WO-2004070050-A2 CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-08-19 WO disclosed