SCHEMBL6182219

SCHEMBL6182219

COCCN1CCC(c2ccc(-c3c[c]ccc3)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.44
SLC18A3 Q16572 2/20 0.43
HRH1 P35367 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
HRH2 P25021 1/20 0.42
KDM1A O60341 1/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4576853 0.80 DRD2 (0.50) DRD2SLC18A3HRH1HRH3KDM1A
SCHEMBL8096432 0.77 DRD2 (0.68) DRD2SLC18A3HRH3KDM1ACARM1
SCHEMBL81936 0.76 DRD2 (0.55) DRD2SLC18A3HRH3KDM1ATLR9
SCHEMBL14320360 0.74 DRD2 (0.54) DRD2SLC18A3HRH1KDM1ATLR9
SCHEMBL22804312 0.74 DRD2 (0.54) DRD2SLC18A3KDM1ACARM1PRMT6
SCHEMBL7534840 0.72 DRD2 (0.69) DRD2CARM1PRMT6
SCHEMBL22804730 0.71 DRD2 (0.50) DRD2SLC18A3HRH1HRH3KDM1A
SCHEMBL3145598 0.71 RAB9A (0.61) HRH1HRH3
SCHEMBL3149207 0.70 LTA4H (0.71) HRH1HRH3HRH2
SCHEMBL1305330 0.70 SLC18A3 (0.58) DRD2SLC18A3HRH1HRH3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537074-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC. (CA) 2005-06-08 EP disclosed
WO-2004022526-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2004-03-18 WO disclosed