SCHEMBL6185512

SCHEMBL6185512

COC(=O)c1ccc2scc(OC)c2c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.43
MET P08581 1/20 0.43
GSK3B P49841 1/20 0.43
LIMK1 P53667 1/20 0.43
DYRK1A Q13627 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
GAA P10253 2/20 0.40
ABL1 P00519 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK4 Q16654 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
KDM4E B2RXH2 3/20 0.37
POLB P06746 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6182352 0.87 ALDH1A1 (0.41) CA12CA1CA2CA7CA9
SCHEMBL7464618 0.87 CLK1 (0.34) CHEK1METGSK3BLIMK1DYRK1A
Hydrochloric Acid SCHEMBL7464629 0.85 ALDH1A1 (0.40) CA12CA1CA2CA7CA9
SCHEMBL7469703 0.79 MTNR1A (0.36) DYRK1AKDM4EALDH1A1MAPTTSHR
SCHEMBL9115645 0.77 GAA (0.43) GAAABL1KDM4EPOLBHPGD
SCHEMBL523584 0.73 ABL1 (0.57) GAAABL1CA12CA1CA2
SCHEMBL7470966 0.72 BACE1 (0.38) CHEK1METGSK3BLIMK1DYRK1A
SCHEMBL9117375 0.72 LMNA (0.39) GSK3BLIMK1DYRK1ACLK4GAA
SCHEMBL7476511 0.71 TSHR (0.40) KDM4EHPGDALDH1A1GLAMAPT
SCHEMBL8135257 0.71 GAA (0.46) GAAABL1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1160244-B1 Isoxazole derivatives and their use as herbicides BAYER AGRICULTURE LTD (GB) 2005-10-19 EP disclosed
EP-0636622-B1 Isoxazole derivatives and their use as herbicides AVENTIS AGRICULTURE LTD (GB) 2002-10-23 EP disclosed
EP-1160244-A1 Isoxazole derivatives and their use as herbicides RHONE-POULENC AGRICULTURE LIMITED (GB) 2001-12-05 EP disclosed
US-5489570-A PRE- OR POST-EMERGENCE RHONE-POULENC AGRICULTURE LIMITED (GB) 1996-02-06 US disclosed
WO-1995025099-A1 2-CYANO-1,3-DIONE DERIVATIVES USEFUL AS HERBICIDES RHONE-POULENC AGRICULTURE LTD. (GB) 1995-09-21 WO disclosed
EP-0636622-A1 Isoxazole derivatives and their use as herbicides RHONE POULENC AGRICULTURE LTD. (GB) 1995-02-01 EP disclosed