SCHEMBL618695

SCHEMBL618695

Cc1nc2ccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)cc2s1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 8/20 0.61
LMNA P02545 7/20 0.61
SMN1; SMN2 Q16637 5/20 0.61
HSD11B1 P28845 1/20 0.60
PKM P14618 1/20 0.59
NOD2 Q9HC29 1/20 0.59
MAPT P10636 2/20 0.53
POLB P06746 1/20 0.53
GAA P10253 1/20 0.53
CDK1 P06493 1/20 0.53
CCNB1 P14635 1/20 0.53
CCNA2 P20248 1/20 0.53
CDK2 P24941 1/20 0.53
CDK7 P50613 1/20 0.53
CCNH P51946 1/20 0.53
CCNA1 P78396 1/20 0.53
ALDH1A1 P00352 3/20 0.53
MAPK1 P28482 1/20 0.52
MEN1 O00255 1/20 0.52
THRB P10828 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4883530 0.91 LMNA (0.61) HTTLMNASMN1; SMN2PKMNOD2
SCHEMBL10089757 0.91 LMNA (0.64) HTTLMNASMN1; SMN2HSD11B1PKM
SCHEMBL27422022 0.83 LMNA (0.63) HTTLMNASMN1; SMN2PKMNOD2
SCHEMBL617881 0.82 LMNA (0.62) HTTLMNASMN1; SMN2HSD11B1PKM
SCHEMBL617597 0.82 HSD11B1 (0.65) HTTLMNAHSD11B1PKMALDH1A1
SCHEMBL3023347 0.81 LMNA (0.73) HTTLMNASMN1; SMN2PKMNOD2
SCHEMBL4875632 0.81 LMNA (0.64) HTTLMNASMN1; SMN2HSD11B1PKM
SCHEMBL13299234 0.78 LMNA (0.82) HTTLMNASMN1; SMN2PKMNOD2
SCHEMBL5348053 0.78 ALPL (0.58) HTTLMNASMN1; SMN2MAPTCDK1
SCHEMBL10089750 0.77 LMNA (0.59) HTTLMNASMN1; SMN2PKMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120041207-A1 Compound STERIX LIMITED (GB) 2012-02-16 US disclosed
US-20120041207-A1 Compound STERIX LIMITED (GB) 2012-02-16 US disclosed
US-20120041207-A1 Compound STERIX LIMITED (GB) 2012-02-16 US disclosed
US-20110009448-A1 Compound STERIX LIMITED 2011-01-13 US disclosed
US-7786152-B2 Compound STERIX LIMITED (GB) 2010-08-31 US disclosed
US-7786152-B2 Compound STERIX LIMITED (GB) 2010-08-31 US disclosed
US-7786152-B2 Compound STERIX LIMITED (GB) 2010-08-31 US disclosed
US-20080114042-A1 Inhibiting 11 beta-hydroxysteroid dehydrogenase (11 beta-HSD); use of sulfonamide-substituted N-heterocyclics including pyrroles, oxazoles, thiazoles, imidazoles and their fused analogs to treat diabetes, obesity, hypertension, arthritis, asthma, osteoporosis, breast cancer STERIX LIMITED (GB) 2008-05-15 US disclosed
US-20080114042-A1 Inhibiting 11 beta-hydroxysteroid dehydrogenase (11 beta-HSD); use of sulfonamide-substituted N-heterocyclics including pyrroles, oxazoles, thiazoles, imidazoles and their fused analogs to treat diabetes, obesity, hypertension, arthritis, asthma, osteoporosis, breast cancer STERIX LIMITED (GB) 2008-05-15 US disclosed
US-20080114042-A1 Inhibiting 11 beta-hydroxysteroid dehydrogenase (11 beta-HSD); use of sulfonamide-substituted N-heterocyclics including pyrroles, oxazoles, thiazoles, imidazoles and their fused analogs to treat diabetes, obesity, hypertension, arthritis, asthma, osteoporosis, breast cancer STERIX LIMITED (GB) 2008-05-15 US disclosed
US-7309715-B2 Compound STERIX LIMITED (GB) 2007-12-18 US disclosed
US-7309715-B2 Compound STERIX LIMITED (GB) 2007-12-18 US disclosed
US-7309715-B2 Compound STERIX LIMITED (GB) 2007-12-18 US disclosed
EP-1556040-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 AND TYPE 2 Sterix Limited (GB) 2005-07-27 EP disclosed
US-20040143124-A1 Compound STERIX LIMITED (GB) 2004-07-22 US disclosed
WO-2004037251-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 AND TYPE 2 STERIX LIMITED (GB) 2004-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080114042-A1 Inhibiting 11 beta-hydroxysteroid dehydrogenase (11 beta-HSD); use of sulfonamide-substituted N-heterocyclics including pyrroles, oxazoles, thiazoles, imidazoles and their fused analogs to treat diabetes, obesity, hypertension, arthritis, asthma, osteoporosis, breast cancer HSD11B1, HSD3B1, HSD11B2 HTT 4116/4885LMNA 4577/4885SMN1; SMN2 3762/4885
US-20110009448-A1 Compound NR4A1, GPR6, PRMT6 HTT 3139/4885LMNA 3102/4885SMN1; SMN2 3761/4885
US-20120041207-A1 Compound NR4A1, GPR6, PRMT6 HTT 3139/4885LMNA 3102/4885SMN1; SMN2 3761/4885
US-20040143124-A1 Compound NR4A1, CBR1, NR2C2 HTT 3836/4885LMNA 2144/4885SMN1; SMN2 3175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.