SCHEMBL6188700

SCHEMBL6188700

CC(C)(C)OC(=O)NC(C)(C)c1cccc(C(=O)c2cc(OC3CCCCO3)ccc2N)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
DHFR P00374 1/20 0.36
BTK Q06187 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 3/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD11B1 P28845 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
ICAM1 P05362 1/20 0.32
SELE P16581 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6188556 0.82 DHFR (0.33) HTTDHFRHSD11B1
SCHEMBL6188956 0.77 GAA (0.46) MEN1KMT2AALDH1A1L3MBTL1LMNA
SCHEMBL6188581 0.76 RECQL (0.40) LMNA
SCHEMBL8205525 0.70 ACACB (0.34) DHFRMEN1KMT2A
SCHEMBL8205526 0.70 NPSR1 (0.35) DHFRMEN1KMT2ANPSR1
SCHEMBL23704909 0.70 RXRA (0.43) HTTMEN1KMT2AALDH1A1L3MBTL1
SCHEMBL8209894 0.70 DHFR (0.38) DHFRMEN1KMT2AHSD11B1L3MBTL1
SCHEMBL28450438 0.69 HPGD (0.44) MEN1KMT2AALDH1A1
SCHEMBL6190860 0.69 DHFR (0.39) DHFRMEN1KMT2AALDH1A1HSD11B1
SCHEMBL6190273 0.68 S1PR3 (0.38) DHFRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-B1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA PHARMACEUTICAL (JP) 2005-11-16 EP disclosed
US-6352982-B1 TREATING DIABETES, OBESITY, OR INVETERATE DIARRHEA IN A MAMMAL WHICH COMPRISES ADMINISTERING AN EFFECTIVE AMOUNT OF A COMPOUND OF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-03-05 US disclosed