SCHEMBL8205526

SCHEMBL8205526

CC(C)(C)OC(=O)NCCCc1cc(OC2CCCCO2)cc(C(=O)c2ccccc2)c1N

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
CNR2 P34972 1/20 0.35
METAP2 P50579 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ATR Q13535 2/20 0.35
CA12 O43570 4/20 0.34
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA9 Q16790 4/20 0.34
SIGMAR1 Q99720 2/20 0.34
DHFR P00374 1/20 0.34
BRD4 O60885 1/20 0.34
ACACB O00763 2/20 0.34
ACACA Q13085 2/20 0.34
IDO1 P14902 1/20 0.33
ADRA2C P18825 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8205525 0.82 ACACB (0.34) MEN1KMT2ADHFRACACBACACA
SCHEMBL8198955 0.78 BRD4 (0.40) SIGMAR1BRD4IDO1
SCHEMBL8199082 0.72 NQO2 (0.44) MEN1KMT2AIDO1
SCHEMBL12635025 0.71 ADRB2 (0.43) MEN1KMT2AATRCA12CA1
SCHEMBL8197947 0.71 IDO1 (0.41) NPSR1MEN1KMT2ACA12CA1
SCHEMBL6188718 0.71 EPHX2 (0.41) MEN1KMT2A
SCHEMBL8211448 0.70 DHFR (0.36) NPSR1ATRCA12CA1CA2
SCHEMBL6188700 0.70 HTT (0.38) NPSR1MEN1KMT2ADHFR
SCHEMBL375762 0.67 MEN1 (0.48) NPSR1METAP2MEN1KMT2ACA12
SCHEMBL11767308 0.67 ELANE (0.52) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 2000-02-16 EP disclosed
WO-1998047882-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-29 WO disclosed