SCHEMBL6189538

SCHEMBL6189538

COc1cc[c]c(-c2ccccc2)c1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 3/20 0.39
PDE4B Q07343 3/20 0.39
PDE4A P27815 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
NFE2L2 Q16236 1/20 0.38
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4024400 0.84 IDO1 (0.40) ALDH1A1IDO1TDO2CA12CA1
SCHEMBL10634123 0.81 ACHE (0.42) ALDH1A1KDM4EHPGDCA12CA1
SCHEMBL7071376 0.81 PDE4B (0.39) ALDH1A1KDM4EHPGDPDE4BPDE4A
SCHEMBL16719798 0.80 TDO2 (0.43) ALDH1A1KDM4EHPGDPDE4BPDE4A
SCHEMBL6681241 0.80 CA12 (0.37) ALDH1A1KDM4EHPGDPDE4BCA12
SCHEMBL9507449 0.80 TUBB4A (0.43) ALDH1A1KDM4EHPGDTUBB4ATUBB
SCHEMBL15623366 0.78 SMN1; SMN2 (0.41) ALDH1A1KDM4EHPGDCA12CA1
SCHEMBL7699767 0.78 KDM4E (0.39) ALDH1A1KDM4EHPGDPDE4BPDE4A
SCHEMBL1274782 0.77 CA1 (0.46) ALDH1A1KDM4EHPGDPDE4BCA12
SCHEMBL9509851 0.76 ALDH1A1 (0.39) ALDH1A1KDM4EHPGDSMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592683-A2 HETEROCYCLYL-3-SULFONYLINDAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2005-11-09 EP disclosed
WO-2004074243-A2 HETEROCYCLYL-3-SULFONYLINDAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2004-09-02 WO disclosed
US-6030975-A ANTAGONIST OF ENDOTHELINS, I.E. INHIBITION OF BINDING WITH RECEPTOR; ANTITUMOR AND -CARCINOGENIC AGENTS; SIDE EFFECT REDUCTION BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
US-5969134-A CARDIOVASCULAR DISORDERS, VASOCONSTRICTION, HYPOTENSIVE AGENTS AND RELEASE OF ENDOTHELINS BASF AKTIENGESELLSCHAFT (DE) 1999-10-19 US disclosed
US-5932730-A Carboxylic acid derivatives, their preparation and use BASF AKTIENGESELLSCHAFT (DE) 1999-08-03 US disclosed
EP-0850222-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 1998-07-01 EP disclosed
WO-1998000402-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1998-01-08 WO disclosed
US-4604383-A ANTICONVULSANTS SOCIETE ANONYME STYLED: SANOFI (FR) 1986-08-05 US disclosed