Morphine

Morphine

SCHEMBL619013

CBr.CN1CC[C@]23c4c5ccc(O)c4O[C@H]2[C@@H](O)C=C[C@H]3[C@H]1C5

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1

The experimentally established mechanism targets of Morphine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 8/20 0.96
OPRD1 P41143 11/20 0.96
OPRK1 P41145 7/20 0.96
MRGPRX2 Q96LB1 4/20 0.96
SLC22A1 O15245 1/20 0.96
ADRA2A P08913 1/20 0.96
ARRB1 P49407 1/20 0.96
ADRB1 P08588 1/20 0.73
PDE4D Q08499 1/20 0.73
PDE3A Q14432 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morphine SCHEMBL7987114 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL13154676 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL13076870 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL8049464 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL13696339 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL24599520 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL2997 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL10820235 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL5183254 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL13695381 0.98 OPRD1 (1.00) OPRD1OPRM1OPRK1MRGPRX2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 194 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240288374-A1 PLASMONIC NANOPARTICLE PLATFORM FOR ANALYTE DETECTION Zymeron Corporation 2024-08-29 US claimed
WO-2024172892-A1 PLASMONIC NANOPARTICLE PLATFORM FOR ANALYTE DETECTION Zymeron Corporation (US) 2024-08-22 WO claimed
US-20230414604-A1 MORPHINE FORMULATIONS FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2023-12-28 US claimed
US-20200345720-A1 MORPHINE FORMULATIONS FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2020-11-05 US claimed
US-20190167665-A1 MORPHINE FORMULATIONS FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2019-06-06 US claimed
US-20160175297-A1 Morphine Formulations FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2016-06-23 US claimed
EP-2968132-A1 INJECTABLE MORPHINE FORMULATIONS Becton Dickinson France S.A.S (FR) 2016-01-20 EP claimed
US-9192608-B2 Morphine formulations BECTON DICKINSON FRANCE S.A.S. (FR) 2015-11-24 US claimed
US-20150246036-A1 Morphine Formulations FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2015-09-03 US claimed
WO-2014153099-A2 METHOD FOR USING EXHALED BREATH TO DETERMINE THE PRESENCE OF DRUG Pulmonary Analytics (US) 2014-09-25 WO claimed
US-20140288454-A1 Method For Using Exhaled Breath to Determine the Presence of Drug Pulmonary Analytics (US) 2014-09-25 US claimed
WO-2014140095-A1 INJECTABLE MORPHINE FORMULATIONS BECTON DICKINSON FRANCE S.A.S. (FR) 2014-09-18 WO claimed
EP-0767663-B1 COMPOSITION COMPRISING MORPHINE, POLYPYRROLIDONE AND A POLYALKYLENEOXIDE ALZA CORP (US) 2002-04-03 EP claimed
EP-0767663-A1 COMPOSITION COMPRISING MORPHINE, POLYPYRROLIDONE AND A POLYALKYLENEOXIDE ALZA CORPORATION (US) 1997-04-16 EP claimed
US-5593695-A Morphine therapy ALZA CORPORATION (US) 1997-01-14 US claimed
WO-1996000066-A1 COMPOSITION COMPRISING MORPHINE, POLYPYRROLIDONE AND A POLYALKYLENEOXIDE ALZA CORPORATION (US) 1996-01-04 WO claimed
US-4126684-A 4-AMINO-3-P-HALOPHENYLBUTYRIC ACIDS AND THEIR DERIVATIVES USED IN THE CONTROL OF NARCOTIC ABUSE CIBA-GEIGY CORPORATION (US) 1978-11-21 US claimed
US-20260060822-A1 BIOENGINEERED SCAFFOLDS FOR VASCULAR GRAFTS AND METHODS OF USE THEREOF UNIV WAKE FOREST HEALTH SCIENCES (US) 2026-03-05 US disclosed
WO-1998031358-A1 d-METHADONE, A NONOPIOID ANALGESIC CORNELL RESEARCH FOUNDATION, INC. (US) 1998-07-23 WO disclosed
US-4126684-A 4-AMINO-3-P-HALOPHENYLBUTYRIC ACIDS AND THEIR DERIVATIVES USED IN THE CONTROL OF NARCOTIC ABUSE CIBA-GEIGY CORPORATION (US) 1978-11-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200345720-A1 MORPHINE FORMULATIONS OPRM1, OPRK1, OPRD1 OPRM1 1/4885OPRD1 3/4885OPRK1 2/4885
US-20190167665-A1 MORPHINE FORMULATIONS OPRM1, OPRK1, OPRD1 OPRM1 1/4885OPRD1 3/4885OPRK1 2/4885
US-20260060822-A1 BIOENGINEERED SCAFFOLDS FOR VASCULAR GRAFTS AND METHODS OF USE THEREOF PFKP, PBK, MYLK OPRM1 4810/4885OPRD1 4518/4885OPRK1 2862/4885
US-20230414604-A1 MORPHINE FORMULATIONS OPRM1, OPRK1, OPRD1 OPRM1 1/4885OPRD1 3/4885OPRK1 2/4885
US-20150246036-A1 Morphine Formulations OPRM1, OPRK1, OPRD1 OPRM1 1/4885OPRD1 3/4885OPRK1 2/4885
US-20160175297-A1 Morphine Formulations OPRM1, OPRK1, OPRD1 OPRM1 1/4885OPRD1 3/4885OPRK1 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.