SCHEMBL6199826

SCHEMBL6199826

O=c1ccn(CCO)c(C(O)c2ccc3ccccc3c2)c1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT2B7 P16662 1/20 0.37
TEAD4 Q15561 1/20 0.36
MAPT P10636 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
ATM Q13315 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC2 Q92769 1/20 0.36
NQO1 P15559 1/20 0.34
TNF P01375 1/20 0.34
HTR1A P08908 1/20 0.34
CYP2D6 P10635 3/20 0.34
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 3/20 0.34
SLC6A3 Q01959 3/20 0.34
KCNH2 Q12809 2/20 0.34
KDM4E B2RXH2 2/20 0.34
AOC3 Q16853 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8850682 0.85 CYP1A2 (0.40) UGT2B7TEAD4MEN1KMT2AHDAC8
SCHEMBL6195293 0.84 KDM4E (0.41) HDAC8HDAC4HDAC2CYP2D6KDM4E
SCHEMBL6199262 0.81 CES2 (0.35) TEAD4MAPTHDAC4SLC6A2SLC6A4
SCHEMBL8850424 0.80 TNF (0.52) TNFCYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6196542 0.80 KMT2A (0.33) TEAD4KMT2ACYP2D6KDM4ETP53
SCHEMBL6196493 0.80 KDM4E (0.34) CYP2D6KDM4ECYP1A2TP53HTT
SCHEMBL6197600 0.80 KDM4E (0.37) TEAD4MAPTKMT2ACYP2D6KDM4E
SCHEMBL6196517 0.80 FPR2 (0.33) TEAD4CYP2D6KDM4ETP53HTT
SCHEMBL6193968 0.78 TSHR (0.47) MAPTMEN1KMT2ANQO1TSHR
SCHEMBL6194701 0.78 MAPK1 (0.39) MEN1KMT2AKDM4EHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0768302-B1 Hydroxypyridinones NOVARTIS AG (CH) 2005-07-06 EP disclosed
US-5688815-A COMPOUNDS FOR REMOVAL OF EXCESS IRON IN MAMMALS CIBA GEIGY CORPORATION (US) 1997-11-18 US disclosed
EP-0768302-A2 Hydroxypyridinones Novartis AG (CH) 1997-04-16 EP disclosed