SCHEMBL6200952

SCHEMBL6200952

Cc1ccc(/C=C\C(=O)c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 1.00
CYP3A4 P08684 3/20 1.00
ALDH1A1 P00352 2/20 1.00
HPGD P15428 1/20 1.00
CYP1B1 Q16678 3/20 0.86
MAOB P27338 6/20 0.75
BCHE P06276 2/20 0.75
LMNA P02545 2/20 0.75
PLIN1 O60240 1/20 0.75
TNFRSF1A P19438 1/20 0.75
ACHE P22303 1/20 0.75
RECQL P46063 1/20 0.75
PLIN5 Q00G26 1/20 0.75
ABHD5 Q8WTS1 1/20 0.75
MAOA P21397 4/20 0.72
RAB9A P51151 3/20 0.72
POLB P06746 1/20 0.72
NFKB1 P19838 2/20 0.71
NFKB2 Q00653 2/20 0.71
RELA Q04206 2/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL76030 1.00 MAPT (1.00) MAPTCYP3A4ALDH1A1HPGDCYP1B1
SCHEMBL5753797 1.00 MAPT (1.00) MAPTCYP3A4ALDH1A1HPGDCYP1B1
SCHEMBL27977352 0.95 MAPT (0.90) MAPTCYP3A4ALDH1A1HPGDCYP1B1
SCHEMBL23789072 0.93 MAPT (0.87) MAPTCYP3A4ALDH1A1HPGDCYP1B1
SCHEMBL7193506 0.93 CYP1B1 (1.00) MAPTCYP3A4ALDH1A1HPGDCYP1B1
SCHEMBL77498 0.93 CYP1B1 (1.00) MAPTCYP3A4ALDH1A1HPGDCYP1B1
SCHEMBL12533800 0.91 MAPT (0.82) MAPTCYP3A4ALDH1A1HPGDCYP1B1
4,4'-Dimethylchalcone SCHEMBL979560 0.90 MAPT (1.00) MAPTCYP3A4ALDH1A1HPGDCYP1B1
4,4'-Dimethylchalcone SCHEMBL979559 0.90 MAPT (1.00) MAPTCYP3A4ALDH1A1HPGDCYP1B1
SCHEMBL9915665 0.90 CYP1B1 (0.91) MAPTCYP3A4ALDH1A1HPGDCYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
US-4261988-A ANTICHOLESTEROL AGENTS USED IN ANIMAL HUSBANDRY BAYER AKTIENGESELLSCHAFT (DE) 1981-04-14 US disclosed