SCHEMBL6201456

SCHEMBL6201456

FC(F)(F)c1cccc(Oc2ccncc2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.58
KDR P35968 1/20 0.58
MAPK14 Q16539 1/20 0.58
TNNI3K Q59H18 1/20 0.58
LTA4H P09960 1/20 0.49
TEAD1 P28347 1/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
ALDH1A1 P00352 2/20 0.48
POLB P06746 2/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.46
MAPT P10636 1/20 0.46
KIF11 P52732 1/20 0.46
P2RY1 P47900 2/20 0.45
TTBK1 Q5TCY1 1/20 0.45
ADORA2A P29274 1/20 0.45
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27579381 0.87 LTA4H (0.59) MAPK14LTA4HTEAD1L3MBTL1ALDH1A1
SCHEMBL9798371 0.87 LTA4H (0.54) LTA4HTEAD1L3MBTL1ALDH1A1POLB
SCHEMBL9546526 0.85 L3MBTL1 (0.55) MAPK14LTA4HTEAD1L3MBTL1ALDH1A1
SCHEMBL14527443 0.81 TLR7 (0.57) BRAFKDRMAPK14TNNI3KL3MBTL1
SCHEMBL694092 0.79 LTA4H (0.49) LTA4HTEAD1L3MBTL1ALDH1A1POLB
SCHEMBL15635197 0.79 PPARG (0.55) MAPK14LTA4HTEAD1L3MBTL1ALDH1A1
SCHEMBL476378 0.79 ALDH1A1 (0.66) LTA4HL3MBTL1ALDH1A1NPSR1MAPT
SCHEMBL13809396 0.79 LTA4H (0.52) MAPK14LTA4HTEAD1L3MBTL1ALDH1A1
SCHEMBL4043144 0.79 LTA4H (0.53) BRAFKDRMAPK14TNNI3KLTA4H
SCHEMBL5542591 0.79 LTA4H (0.52) MAPK14LTA4HTEAD1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208104-B1 TRICYCLIC INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASES AGOURON PHARMA (US) 2005-01-19 EP disclosed
US-4411904-A Diphenylpropanamines, compositions thereof and use thereof WARNER-LAMBERT COMPANY (US) 1983-10-25 US disclosed
US-4364954-A NEUROLEPTIC AGENT WARNER-LAMBERT COMPANY (US) 1982-12-21 US disclosed
US-4292321-A 1,3,8-Triazaspirodecane-4-ones, pharmaceutical compositions thereof and method of use thereof WARNER-LAMBERT COMPANY (US) 1981-09-29 US disclosed
US-4218456-A 1-(4-Fluorophenyl)-4-(1,2,3,6-tetrahydro-4-phenoxy-1-pyridinyl)-butanones WARNER-LAMBERT COMPANY (US) 1980-08-19 US disclosed