SCHEMBL6203751

SCHEMBL6203751

O=C(c1cccnc1)C(Cc1ccco1)c1ccc(Cl)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 7/20 0.42
KDM4E B2RXH2 3/20 0.42
LMNA P02545 3/20 0.42
PKM P14618 2/20 0.42
MAPT P10636 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
USP2 O75604 1/20 0.41
RAB9A P51151 2/20 0.40
POLB P06746 2/20 0.40
NPC1 O15118 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
HPGD P15428 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204706 0.83 NPC1 (0.46) ALDH1A1KDM4ELMNAPKMMAPT
SCHEMBL6202785 0.82 NPC1 (0.46) TDP1ALDH1A1KDM4ELMNAPKM
SCHEMBL6199987 0.81 RAB9A (0.43) ALDH1A1KDM4ELMNAPKMMAPT
SCHEMBL9877648 0.81 ALDH1A1 (0.48) ALDH1A1KDM4ELMNAPKMMAPT
SCHEMBL9878025 0.79 ALDH1A1 (0.46) MAPK1ALDH1A1KDM4ELMNAPKM
SCHEMBL9877329 0.78 ALDH1A1 (0.46) TDP1ALDH1A1KDM4ELMNAPKM
SCHEMBL10448844 0.78 ALDH1A1 (0.48) TDP1ALDH1A1KDM4ELMNAPKM
SCHEMBL11094696 0.78 ALDH1A1 (0.48) TDP1ALDH1A1KDM4ELMNAPKM
SCHEMBL11094694 0.78 ALDH1A1 (0.48) TDP1ALDH1A1KDM4ELMNAPKM
SCHEMBL11096738 0.77 ALDH1A1 (0.45) MAPK1TDP1ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
EP-0117485-A2 Pyridine, pyrazine and pyrimidine derivatives and their use as fungicides F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-09-05 EP disclosed