SCHEMBL6204294

SCHEMBL6204294

O=C(NC(=O)C1CCCNC1)c1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
HTT P42858 1/20 0.51
GPR6 P46095 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
CDK2AP1 O14519 1/20 0.43
CHEK1 O14757 1/20 0.43
TSHR P16473 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
LMNA P02545 1/20 0.43
HIF1A Q16665 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203700 0.84 KDM4E (0.45) ALDH1A1SMN1; SMN2CDK2AP1CHEK1TSHR
SCHEMBL7241178 0.83 CHRNB2 (0.48) ALDH1A1SMN1; SMN2CHRNB2CHRNA4TSHR
SCHEMBL6204321 0.82 HDAC1 (0.48) HDAC1HDAC6
SCHEMBL6203532 0.82 HDAC1 (0.48) HDAC1HDAC6
SCHEMBL6203499 0.82 HDAC1 (0.48) HDAC1HDAC6
Hydrochloric Acid SCHEMBL15648258 0.82 CHRNB2 (0.47) ALDH1A1SMN1; SMN2CHRNB2CHRNA4TSHR
SCHEMBL14490487 0.80 HTT (0.53) ALDH1A1HTTGPR6HDAC1HDAC6
SCHEMBL29542503 0.80 DYRK1B (0.56)
SCHEMBL6204397 0.79 SMYD3 (0.46)
SCHEMBL6204513 0.79 SMYD3 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494672-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2005-01-12 EP disclosed
WO-2003086398-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-10-23 WO disclosed