SCHEMBL6204513

SCHEMBL6204513

Cc1cncc(C(=O)NC(=O)[C@H]2CCCNC2)c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 3/20 0.46
ACKR3 P25106 7/20 0.41
ATM Q13315 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
ULK1 O75385 1/20 0.39
WNT1 P04628 3/20 0.39
GSK3B P49841 3/20 0.39
DYRK1A Q13627 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204397 1.00 SMYD3 (0.46) SMYD3ACKR3ATMHCAR2ULK1
SCHEMBL6204294 0.79 ALDH1A1 (0.51)
SCHEMBL6204321 0.79 HDAC1 (0.48) WNT1GSK3BDYRK1A
SCHEMBL6203499 0.79 HDAC1 (0.48) WNT1GSK3BDYRK1A
SCHEMBL6203532 0.79 HDAC1 (0.48) WNT1GSK3BDYRK1A
SCHEMBL6203700 0.78 KDM4E (0.45) ATMULK1
SCHEMBL6277414 0.77 SMYD3 (0.47) SMYD3ACKR3ATMHCAR2ULK1
SCHEMBL6371533 0.73 HDAC1 (0.50) ACKR3
SCHEMBL3879671 0.73 NPC1 (0.47) ATM
SCHEMBL3877272 0.72 TAS1R3 (0.45) ULK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494672-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2005-01-12 EP disclosed
WO-2003086398-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-10-23 WO disclosed