SCHEMBL6203700

SCHEMBL6203700

O=C(NC(=O)C1CCCNC1)c1ccncc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
CYP2D6 P10635 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
ULK1 O75385 1/20 0.43
SLC6A1 P30531 2/20 0.42
SLC6A11 P48066 1/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SLC6A13 Q9NSD5 1/20 0.42
AKT1 P31749 4/20 0.42
AKT2 P31751 2/20 0.42
AKT3 Q9Y243 2/20 0.42
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
PBK Q96KB5 1/20 0.41
TNKS O95271 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204294 0.84 ALDH1A1 (0.51) TSHRLMNASMN1; SMN2MAPTALDH1A1
SCHEMBL3879671 0.83 NPC1 (0.47) KDM4ECYP2D6SLC6A1SLC6A11TSHR
SCHEMBL6201040 0.82 ALDH1A1 (0.47) KDM4ECYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL1552756 0.80 ULK1 (0.56) CYP2D6CYP3A4ULK1TSHRLMNA
SCHEMBL6204321 0.79 HDAC1 (0.48)
SCHEMBL6203499 0.79 HDAC1 (0.48)
SCHEMBL6203532 0.79 HDAC1 (0.48)
SCHEMBL6204513 0.78 SMYD3 (0.46) ULK1ATM
SCHEMBL6204397 0.78 SMYD3 (0.46) ULK1ATM
SCHEMBL3877272 0.77 TAS1R3 (0.45) ULK1SLC6A1SLC6A11TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494672-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2005-01-12 EP disclosed
WO-2003086398-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-10-23 WO disclosed