SCHEMBL6203734

SCHEMBL6203734

O=C(Cc1ccncc1)c1ccncc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
PLOD2 O00469 2/20 0.55
PLOD3 O60568 2/20 0.55
PLOD1 Q02809 2/20 0.55
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 2/20 0.55
CYP2C19 P33261 2/20 0.55
CYP2C9 P11712 1/20 0.55
HPGD P15428 1/20 0.55
HIF1A Q16665 1/20 0.55
NAPRT Q6XQN6 1/20 0.50
KDM4E B2RXH2 1/20 0.48
MPO P05164 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP19A1 P11511 3/20 0.47
MAPT P10636 3/20 0.47
L3MBTL1 Q9Y468 3/20 0.47
GAA P10253 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1157353 0.90 ALDH1A1 (0.66) ALDH1A1PLOD2PLOD3PLOD1CYP1A2
SCHEMBL1515846 0.90 ALDH1A1 (0.66) ALDH1A1PLOD2PLOD3PLOD1CYP1A2
SCHEMBL6775249 0.88 NPC1 (0.62) ALDH1A1PLOD2PLOD3PLOD1CYP1A2
SCHEMBL2645324 0.86 LTA4H (0.58) ALDH1A1PLOD2CYP3A4MAPTL3MBTL1
SCHEMBL4102938 0.86 L3MBTL1 (0.68) CYP3A4KDM4EMAPTL3MBTL1NPC1
SCHEMBL6101952 0.86 RAB9A (0.66) ALDH1A1PLOD2PLOD3PLOD1CYP1A2
SCHEMBL1395223 0.86 RAB9A (0.64) ALDH1A1PLOD2PLOD3PLOD1CYP1A2
SCHEMBL1993655 0.86 L3MBTL1 (0.58) ALDH1A1PLOD2PLOD3PLOD1CYP1A2
SCHEMBL7433779 0.86 LMNA (0.58) ALDH1A1KDM4EMAPTL3MBTL1SRD5A2
SCHEMBL2512740 0.86 RAB9A (0.64) CYP1A2CYP3A4CYP2D6CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884030-B Improved labeling of nucleophiles using bipyridines 安捷伦科技有限公司 2022-06-28 CN disclosed
US-20210333269-A1 Kits for Using Bispyridines to Improve Labeling of Nucleophiles AGILENT TECHNOLOGIES, INC. (US) 2021-10-28 US disclosed
US-11092595-B2 Use of bispyridines to improve labeling of nucleophiles AGILENT TECHNOLOGIES, INC. (US) 2021-08-17 US disclosed
US-20190041384-A1 USE OF BISPYRIDINES TO IMPROVE LABELING OF NUCLEOPHILES PROZYME, INC. 2019-02-07 US disclosed
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
US-6855710-B2 Substituted indolines with an inhibitory effect on various kinases and complexes of CDKs BOEHRINGER INGELHEIM PHARMA KG (DE) 2005-02-15 US disclosed
US-20040058978-A1 Novel substituted indolines with an inhibitory effect on various kinases and complexes of CDKs BOEHRINGER INGELHEIM PHARMA KG (DE) 2004-03-25 US disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190041384-A1 USE OF BISPYRIDINES TO IMPROVE LABELING OF NUCLEOPHILES PTMS, BTD, DPYD ALDH1A1 633/4885PLOD2 1699/4885PLOD3 3241/4885
US-11092595-B2 Use of bispyridines to improve labeling of nucleophiles PTMS, BTD, DPYD ALDH1A1 633/4885PLOD2 1699/4885PLOD3 3241/4885
US-20210333269-A1 Kits for Using Bispyridines to Improve Labeling of Nucleophiles DPYD, UNG, BTD ALDH1A1 576/4885PLOD2 1613/4885PLOD3 3022/4885
US-20040058978-A1 Novel substituted indolines with an inhibitory effect on various kinases and complexes of CDKs CDK1, CDK2, CDK3 ALDH1A1 1810/4885PLOD2 4746/4885PLOD3 4849/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.