SCHEMBL6203848

SCHEMBL6203848

O=C(CCc1ccc(Cl)cc1)c1ccc(F)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.51
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
SLC5A1 P13866 1/20 0.47
SLC5A2 P31639 1/20 0.47
MDM2 Q00987 2/20 0.46
ACKR3 P25106 2/20 0.45
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
PLAAT3 P53816 1/20 0.43
PLAAT5 Q96KN8 1/20 0.43
PLAAT2 Q9NWW9 1/20 0.43
PLAAT4 Q9UL19 1/20 0.43
CNR1 P21554 1/20 0.43
POLB P06746 1/20 0.43
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
GPR84 Q9NQS5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203033 0.91 SLC5A1 (0.55) RAB9ANPC1CES2CES1SLC5A1
SCHEMBL6161424 0.85 CES2 (0.47) RAB9ACES2CES1SLC5A1SLC5A2
SCHEMBL13988809 0.82 MEN1 (0.48) RAB9ANPC1SLC5A1SLC5A2PLAAT3
SCHEMBL656917 0.81 CYP19A1 (0.51) DRD2RAB9ANPC1CES2CES1
SCHEMBL24511805 0.80 MCHR1 (0.47) CYP11B1CYP11B2
SCHEMBL657632 0.78 TP53 (0.59) DRD2RAB9ANPC1SLC5A1SLC5A2
SCHEMBL6202254 0.78 TP53 (0.59) DRD2RAB9ANPC1SLC5A1SLC5A2
SCHEMBL3739418 0.78 ALDH1A1 (0.61) RAB9APLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL959448 0.77 CES2 (0.57) DRD2RAB9ANPC1CES2CES1
SCHEMBL656153 0.76 GPR84 (0.55) DRD2RAB9ANPC1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed